TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 1.60nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 3.70nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory activity of the compound against cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibitory activity of the compound against cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibitory activity of the compound against cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibitory activity of the compound against cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibitory activity of the compound against ChymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Binding affinity of the compound towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity of the compound towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity of the compound towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Cytotoxic activity in rat liver Huh-7 cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Purdue Pharma Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 150nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 154nMAssay Description:Inhibitory activity of the compound against cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
Affinity DataKi: 176nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity of the compound towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity of the compound towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity of the compound towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibitory activity of the compound against HCV protease using replicon assay in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 229nMAssay Description:Inhibitory activity of the compound against cathepsin KMore data for this Ligand-Target Pair