Affinity DataKi: 0.110nMAssay Description:Displacement of [3H] labeled-N-(4-Fluorophenyl)-3-(4-(4-(2-hydroxypropan-2-yl)-6-(trifluoromethyl)pyridin-3-yl)phenyl)oxetane-3-carboxamide from huma...More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H] labeled-N-(4-Fluorophenyl)-3-(4-(4-(2-hydroxypropan-2-yl)-6-(trifluoromethyl)pyridin-3-yl)phenyl)oxetane-3-carboxamide from huma...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 54.4nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 148nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 161nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Displacement of radiolabeled PDBU from PKC in rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+4nMAssay Description:Purified SOD from bovine brain (20 μl) was incubated (37°C, 60 min) with Aβ25-37, Aβ29-33 or Aβ1-40 (20 μl, 5 μM) follo...More data for this Ligand-Target Pair
Affinity DataKi: 1.32E+4nMAssay Description:Purified SOD from bovine brain (20 μl) was incubated (37°C, 60 min) with Aβ25-37, Aβ29-33 or Aβ1-40 (20 μl, 5 μM) follo...More data for this Ligand-Target Pair
Affinity DataKi: 1.44E+4nMAssay Description:Purified SOD from bovine brain (20 μl) was incubated (37°C, 60 min) with Aβ25-37, Aβ29-33 or Aβ1-40 (20 μl, 5 μM) follo...More data for this Ligand-Target Pair
Affinity DataKi: 5.70E+4nMAssay Description:Competitive inhibition of SARS CoV-2 main protease using varying concentrations of DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by Dixon plot anal...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of IDO1 in IFNgamma/LPS stimulated human whole blood assessed as unbound concentration using kynurenine/tryptophan as substrate preincubat...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of IDO1 in IFNgamma/LPS stimulated human whole blood assessed as unbound concentration using kynurenine/tryptophan as substrate preincubat...More data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of recombinant Jak2 (unknown origin) using biotinylated synthetic peptide substrate by homogeneous time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMpH: 7.5Assay Description:Recombinant human NQO1 was obtained from Sigma and diluted in 50 mM phosphate buffer to give an absorbance of 0.1 at 550 nm; 5 uL of this solution wa...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant Jak2 (unknown origin) using biotinylated synthetic peptide substrate by homogeneous time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Inhibition of IDO1 in IFNgamma/LPS stimulated human whole blood assessed as unbound concentration using kynurenine/tryptophan as substrate preincubat...More data for this Ligand-Target Pair