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Found 45 with Last Name = 'wong' and Initial = 'ecn'
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for in vitro potency against Angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 7.13-7.17More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 8.08-8.22More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 8.70-8.83More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50237727(CHEMBL4060938)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50177595((2S)-5-amino-2-{[(2S)-1-{[(4R,7S,10S,13S,16R)-13-[...)
Affinity DataIC50:  372nMAssay Description:Compound was evaluated for OT receptor affinity by displacement of [3H]OT from binding sites in uterine tissue taken from nonlabor pregnant womenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249034(CHEMBL4077729)
Affinity DataIC50:  2.42E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249036(CHEMBL4066742)
Affinity DataIC50:  3.38E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249039(CHEMBL4101998)
Affinity DataIC50:  4.24E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249038(CHEMBL1409841)
Affinity DataIC50:  4.54E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249041(CHEMBL4081253)
Affinity DataIC50:  4.96E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249040(CHEMBL4080320)
Affinity DataIC50:  5.95E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249037(CHEMBL4104553)
Affinity DataIC50:  6.41E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249035(CHEMBL4094266)
Affinity DataIC50:  6.75E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in CHO cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluores...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249033(CHEMBL4078657)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataEC50:  0.126nMAssay Description:Compound was evaluated for in vitro potency against AT1 receptor in isolated rabbit aorta; value ranges from 7.91-7.97More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataEC50:  0.158nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataEC50:  0.100nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 10.1-10.7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataEC50:  0.0794nMAssay Description:Compound was evaluated for in vitro potency against Angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 5.53-5.69More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataEC50:  0.126nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 8.27-8.70More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataEC50:  8nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataEC50:  0.158nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataEC50:  0.100nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human OTR expressed in HEK293 cell membranes induction of IP1 accumulation at 0.1 to 10 uM measured after 1 hr by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataEC50:  0.0794nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cell membranes assessed as inhibition of OT-induced increase in Ca2+ flux preincubated for 5 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed