Report error Found 195 Enz. Inhib. hit(s) with all data for entry = 50012236
Affinity DataKi: 0.263nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of human CA9 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of human CA9 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibition of human CA1 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Displacement of [3H]-NECA from human A2A receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Inhibition of human CA9 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 183nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 194nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 205nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibition of human CA1 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 279nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 283nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 303nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 319nMAssay Description:Inhibition of human CA9 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 341nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 358nMAssay Description:Inhibition of human CA12 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 367nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped- flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
Affinity DataKi: 395nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair