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Found 6 Enz. Inhib. hit(s) with Target = 'Arginase-1' and Ligand = 'BDBM50230418'
TargetArginase-1(Bos taurus)
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of bovine liver arginaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails PubMedMMDB

TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)
Affinity DataIC50:  3.60E+3nMAssay Description:Binding affinity to human ARG1 assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails PubMedMMDB

TargetArginase-1(Rattus norvegicus)
Oncoarendi Therapeutics

Curated by ChEMBL
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetArginase-1(Rattus norvegicus)
Oncoarendi Therapeutics

Curated by ChEMBL
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of rat ARG1More data for this Ligand-Target Pair
In DepthDetails PubMedMMDB

TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)
Affinity DataKd:  3.60E+3nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB