Affinity DataIC50: 59nMAssay Description:Inhibition of CYP27A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Rattus norvegicus)
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of CYP24A1 in rat kidney mitochondriaMore data for this Ligand-Target Pair
Affinity DataIC50: 4.33E+3nMAssay Description:Inhibition of CYP27A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 5.08E+3nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.34E+3nMAssay Description:Inhibition of CYP27A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.69E+3nMAssay Description:Inhibition of CYP27A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.23E+3nMAssay Description:Inhibition of CYP27A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Rattus norvegicus)
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP24A1 in rat kidney mitochondriaMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 3.43E+5nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataIC50: 4.80E+5nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair