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Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50033388
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344327(2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]py...)
Affinity DataIC50:  55nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344329(2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]py...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344325(4-(6-chloropyridazin-3-yl)-2-isopropyl-7-methoxypy...)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344321(2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]py...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344314(CHEMBL1779432 | rac-2-Benzyl-4a-methyl-4,4a,5,6-te...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344318(CHEMBL1779436 | rac-9-Benzyl-1-isopropyl-6a,9,10b,...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344326(6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-4-y...)
Affinity DataIC50:  2.58E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344328(6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-4-y...)
Affinity DataIC50:  2.61E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344326(6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-4-y...)
Affinity DataIC50:  2.75E+3nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344315(5,6-Dihydro-2H-1,2,7,7a-tetraaza-benzo[c]fluoren-3...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344306((R)-6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-5-m...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50240404((Ibudilast)1-(2-Isopropyl-pyrazolo[1,5-a]pyridin-3...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344327(2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]py...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344311(CHEMBL1779429 | rac-4,4a,5,6-Tetrahydro-2H-1,2,7,7...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344314(CHEMBL1779432 | rac-2-Benzyl-4a-methyl-4,4a,5,6-te...)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344305(CHEMBL1779335 | rac-6-(2-isopropylpyrazolo[1,5-a]p...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344312(CHEMBL1779430 | rac-2-Benzyl-4,4a,5,6-tetrahydro-2...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344306((R)-6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-5-m...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344313(CHEMBL1779431 | rac-4a-Methyl-4,4a,5,6-tetrahydro-...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344307((S)-6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-5-m...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344316(2-Benzyl-5,6-dihydro-2H-1,2,7,7a-tetraaza-benzo[c]...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344319(2-benzyl-6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344320(6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-3-y...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344306((R)-6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-5-m...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344312(CHEMBL1779430 | rac-2-Benzyl-4,4a,5,6-tetrahydro-2...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344329(2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]py...)
Affinity DataIC50:  2.89E+4nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344322(3-(6-chloropyridazin-3-yl)-2-isopropylpyrazolo[1,5...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344313(CHEMBL1779431 | rac-4a-Methyl-4,4a,5,6-tetrahydro-...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344329(2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]py...)
Affinity DataIC50:  3.35E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344317(CHEMBL1779435 | rac-1-Isopropyl-6a,9-dihydro-6H,7H...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344328(6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-4-y...)
Affinity DataIC50:  3.96E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344308(6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-4,5-dih...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344327(2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]py...)
Affinity DataIC50:  4.15E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344305(CHEMBL1779335 | rac-6-(2-isopropylpyrazolo[1,5-a]p...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344322(3-(6-chloropyridazin-3-yl)-2-isopropylpyrazolo[1,5...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344316(2-Benzyl-5,6-dihydro-2H-1,2,7,7a-tetraaza-benzo[c]...)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344309(6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)pyridazi...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344315(5,6-Dihydro-2H-1,2,7,7a-tetraaza-benzo[c]fluoren-3...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344308(6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-4,5-dih...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344309(6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)pyridazi...)
Affinity DataIC50:  7.90E+4nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344305(CHEMBL1779335 | rac-6-(2-isopropylpyrazolo[1,5-a]p...)
Affinity DataIC50:  8.90E+4nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344326(6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-4-y...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50240404((Ibudilast)1-(2-Isopropyl-pyrazolo[1,5-a]pyridin-3...)
Affinity DataIC50:  1.03E+5nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344308(6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-4,5-dih...)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344309(6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)pyridazi...)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344324(2-isopropyl-3-(6-methoxypyridazin-3-yl)pyrazolo[1,...)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344311(CHEMBL1779429 | rac-4,4a,5,6-Tetrahydro-2H-1,2,7,7...)
Affinity DataIC50:  1.45E+5nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344315(5,6-Dihydro-2H-1,2,7,7a-tetraaza-benzo[c]fluoren-3...)
Affinity DataIC50:  1.56E+5nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344311(CHEMBL1779429 | rac-4,4a,5,6-Tetrahydro-2H-1,2,7,7...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344317(CHEMBL1779435 | rac-1-Isopropyl-6a,9-dihydro-6H,7H...)
Affinity DataIC50:  2.10E+5nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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