Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50039559
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380022BDBM50380022(CHEMBL2012509)
Affinity DataIC50: 4.60nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380014BDBM50380014(CHEMBL2012500)
Affinity DataIC50: 6.40nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380018BDBM50380018(CHEMBL2012505)
Affinity DataIC50: 8.10nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380023BDBM50380023(CHEMBL2012510)
Affinity DataIC50: 8.60nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380004BDBM50380004(CHEMBL2012489)
Affinity DataIC50: 8.80nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380012BDBM50380012(CHEMBL2012497)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380006BDBM50380006(CHEMBL2012491)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380019BDBM50380019(CHEMBL2012506)
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380009BDBM50380009(CHEMBL2012494)
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380017BDBM50380017(CHEMBL2012503)
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380011BDBM50380011(CHEMBL2012496)
Affinity DataIC50: 21nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380005BDBM50380005(CHEMBL2012490)
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380003BDBM50380003(CHEMBL2012488)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380007BDBM50380007(CHEMBL2012492)
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380013BDBM50380013(CHEMBL2012499)
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380008BDBM50380008(CHEMBL2012493)
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380015BDBM50380015(CHEMBL2012501)
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380016BDBM50380016(CHEMBL2012502)
Affinity DataIC50: 35nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380010BDBM50380010(CHEMBL2012495)
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380021BDBM50380021(CHEMBL2012508)
Affinity DataIC50: 49nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380024BDBM50380024(CHEMBL2012511)
Affinity DataIC50: 64nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380002BDBM50380002(CHEMBL2012487)
Affinity DataIC50: 225nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380020BDBM50380020(CHEMBL2012507)
Affinity DataIC50: 451nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380001BDBM50380001(CHEMBL2012498)
Affinity DataIC50: 513nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed