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Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50049322
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239006(CHEMBL4060481)
Affinity DataIC50:  29nMAssay Description:Inhibition of DRAK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  250nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50:  330nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238997(CHEMBL4076100)
Affinity DataIC50:  410nMAssay Description:In vitro inhibitory activity against monkey (Callithrix jacchus) plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAngiopoietin-1 receptor(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  510nMAssay Description:Inhibition of human TEKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238996(CHEMBL4099371)
Affinity DataIC50:  690nMAssay Description:In vitro inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAurora kinase A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  850nMAssay Description:In vitro inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAngiopoietin-1 receptor(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  950nMAssay Description:Inhibition of human TEKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238998(CHEMBL4103220)
Affinity DataIC50:  960nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238995(CHEMBL4072438)
Affinity DataIC50:  990nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAurora kinase A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of human AURORA-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238999(CHEMBL4072264)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of hog man plasma renin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239011(CHEMBL4074827)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50024284(CHEMBL3334979)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50024284(CHEMBL3334979)
Affinity DataIC50:  1.72E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase ITK/TSK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of human ITKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 9(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  2.16E+3nMAssay Description:Inhibition of human CDK9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase ITK/TSK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  2.19E+3nMAssay Description:Inhibition of human ITKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeath-associated protein kinase 3(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239003(CHEMBL4101141)
Affinity DataIC50:  2.44E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 6(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  2.44E+3nMAssay Description:Inhibition of human CDK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 4(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  2.82E+3nMAssay Description:Inhibition of human CDK4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase Blk(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  2.88E+3nMAssay Description:Inhibition of human BLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase Blk(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of human BLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeath-associated protein kinase 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  3.07E+3nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50036932(CHEMBL1478023 | US11866416, Compound SN-II-118)
Affinity DataIC50:  3.08E+3nMAssay Description:Compound was tested for the inhibitory constant for mouse kidney cytidine deaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238984(CHEMBL2253274)
Affinity DataIC50:  3.11E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238986(CHEMBL2253275)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239009(CHEMBL4073831)
Affinity DataIC50:  3.66E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase JAK3(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  4.26E+3nMAssay Description:Inhibition of human JAK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  4.63E+3nMAssay Description:Inhibition of human SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase BTK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rat plasma renin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase BTK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  5.03E+3nMAssay Description:In vitro inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase Blk(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50:  5.26E+3nMAssay Description:Inhibition of human BLKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibitory activity against the thymidylate synthase in the Permeabilized L1210 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239013(CHEMBL4101308)
Affinity DataIC50:  5.37E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  5.81E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  5.85E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase BTK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  6.02E+3nMAssay Description:Inhibition of human BTKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50:  6.23E+3nMAssay Description:Inhibition of human IKKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeath-associated protein kinase 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  6.34E+3nMAssay Description:Compound was tested for the inhibitory constant for adenosine deaminase (ADA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238985(CHEMBL4093574)
Affinity DataIC50:  6.65E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239002(CHEMBL4105654)
Affinity DataIC50:  7.16E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238994(CHEMBL4095019)
Affinity DataIC50:  7.26E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50:  8.84E+3nMAssay Description:Inhibition of human CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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