Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50002632
TargetMuscarinic acetylcholine receptor M1(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50460765(CHEMBL4229203)
Affinity DataEC50:  210nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M1 expressed in CHO cells assessed as potentiation of acetylcholine-induced...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50313638(1-(4-methoxybenzyl)-4-oxo-1,4-dihydroquinoline-3-c...)
Affinity DataEC50:  823nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M1 expressed in CHO-NFAT cells assessed as potentiation of acetylcholine-in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50460765(CHEMBL4229203)
Affinity DataEC50:  4.80E+3nMAssay Description:Allosteric agonist at human muscarinic acetylcholine receptor M1 expressed in CHO cells assessed as induction of calcium mobilization after 2.5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed