Compile Data Set for Download or QSAR
maximum 50k data
Found 74 Enz. Inhib. hit(s) with all data for entry = 756
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289421(5-(2-cyclopropyl-1-(3-morpholinobicyclo[1.1.1]pent...)
Affinity DataKd:  11.4nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289422(US10093664, Example 2)
Affinity DataKd:  13nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289423(5-(2-isopropyl-1-(3-morpholinobicyclo[1.1.1]pentan...)
Affinity DataKd:  11nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289424(US10093664, Example 4)
Affinity DataKd:  8.30nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289425((R)-(4-(6-amino-5-(trifluoromethyl)pyridin-3-yl)-1...)
Affinity DataKd:  2.30nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289426( (R)-1-(4-(6-amino-5-(trifluoromethyl)pyridin-3-yl...)
Affinity DataKd:  0.740nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289427((R)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  45nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289428((S)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289429((S)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  0.310nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289430(5-(1-isopropyl-5-(3-morpholinobicyclo[1.1.1]pentan...)
Affinity DataKd:  15nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289431(5-(2-cyclopropyl-1-(3-(4-methylpiperazin-1-yl)bicy...)
Affinity DataKd:  20nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289432(US10093664, Example 13)
Affinity DataKd:  32nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289433(5-(1-(3-(1,4-oxazepan-4-yl)bicyclo[1.1.1]pentan-1-...)
Affinity DataKd:  47nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289434(5-(2-cyclopropyl-1-(3-(4-(2,2,2-trifluoroethyl)pip...)
Affinity DataKd:  18nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289435(5-(2-cyclopropyl-1-(3-(4-(methylsulfonyl)piperazin...)
Affinity DataKd:  24nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289436(5-(2-cyclopropyl-1-(3-(4-(2-fluoroethyl)piperazin-...)
Affinity DataKd:  6.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289437(4-(3-(2-cyclopropyl-4-(3-(trifluoromethyl)-1H-pyrr...)
Affinity DataKd:  1.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289438(5-(2-cyclopropyl-1-(3-(piperidin-1-yl)bicyclo[1.1....)
Affinity DataKd:  14nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289439(4-(3-(2-cyclopropyl-4-(1H-pyrrolo[3,2-b]pyridin-6-...)
Affinity DataKd:  7.50E+3nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289440(4-(3-(2-cyclopropyl-4-(1-(2-fluoroethyl)-H-pyrrolo...)
Affinity DataKd:  330nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289441(4-(3-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl)...)
Affinity DataKd:  9.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289442(1-(3-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl)...)
Affinity DataKd:  17nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289443(5-(2-cyclopropyl-1-(3-((2-methoxyethyl)(methyl)ami...)
Affinity DataKd:  6.80nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289444(5-(1-(3-(bis(2-methoxyethyl)amino)bicyclo[1.1.1]pe...)
Affinity DataKd:  6.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289445(1-(3-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl)...)
Affinity DataKd:  7nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289446(5-(2-cyclopropyl-1-(3-(oxazol-5-yl)bicyclo[1.1.1]p...)
Affinity DataKd:  29nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289447(4-(3-(2-isopropyl-4-(1-(1-(pyridin-2-yl)ethyl)-1H-...)
Affinity DataKd:  2.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289448(1-(4-(6-amino-5- (trifluoromethoxy)- pyridin-3-yl)...)
Affinity DataKd:  20nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289449(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  390nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289454(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  170nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289455(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  6.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289456((S)-1-(4-(6-amino-5- (trifluoromethyl)- pyridin-3-...)
Affinity DataKd:  9.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289457(5-(2-(cyclopropyl- methyl)-1-(3-morpho- linobicycl...)
Affinity DataKd:  29nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289458(5-(2-(cyclopropyl- methyl)-1-(3-morpho- linobicycl...)
Affinity DataKd:  7.20nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289459(5-(2-(cyclopropyl- methyl)-1-(3-morpho- linobicycl...)
Affinity DataKd:  22nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289460(5-(2-cyclopropyl-1-(3- morpholinobicyclo- [1.1.1]p...)
Affinity DataKd:  19nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289461(3-(difluoromethoxy)-5- (2-isopropyl-1-(3- morpholi...)
Affinity DataKd:  19nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289463(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  210nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289464(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  66nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289465(3-(difluoromethoxy)-5- (1-(3-morpholino- bicyclo[1...)
Affinity DataKd:  82nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289466(5-(2-(cyclopropyl- methyl)-1-(3-(4- methylpiperazi...)
Affinity DataKd:  3.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289467(5-(2-cyclobutyl-1-(3- morpholinobicyclo- [1.1.1]pe...)
Affinity DataKd:  32nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289468(5-(2-cyclopentyl-1-(3- morpholinobicyclo- [1.1.1]p...)
Affinity DataKd:  53nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289469(5-(2-isobutyl-1-(3- morpholinobicyclo- [1.1.1]pent...)
Affinity DataKd:  15nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289470(3-(difluoromethoxy)-5- (2-isobutyl-1-(3- morpholin...)
Affinity DataKd:  29nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289471(5-(2-isobutyl-1-(3- morpholinobicyclo- [1.1.1]pent...)
Affinity DataKd:  6nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289472(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  13nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289473(5-(2-(sec-butyl)-1-(3- morpholinobicyclo- [1.1.1]p...)
Affinity DataKd:  8.60nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289474(5-(2-(sec-butyl)-1-(3- morpholinobicyclo- [1.1.1]p...)
Affinity DataKd:  9.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System

US Patent
LigandPNGBDBM289473(5-(2-(sec-butyl)-1-(3- morpholinobicyclo- [1.1.1]p...)
Affinity DataKd:  21nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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