Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 756
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289495BDBM289495(US10093664, Example 67 | 1-(4-(6-amino-5-(tri- flu...)
Affinity DataKd:  0.110nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289483BDBM289483(US10093664, Example 59 | 1-(4-(6-amino-5- (trifluo...)
Affinity DataKd:  0.290nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289429BDBM289429(US10093664, Example 10 | (S)-1-(4-(6-amino-5-(trif...)
Affinity DataKd:  0.310nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289505BDBM289505(US10093664, Example 69a | 1-(4-(6-amino-5-(tri- fl...)
Affinity DataKd:  0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289428BDBM289428(US10093664, Example 8a | (S)-1-(4-(6-amino-5-(trif...)
Affinity DataKd:  0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289481BDBM289481(US10093664, Example 57 | US10093664, Example 62 | ...)
Affinity DataKd:  0.620nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289426BDBM289426(US10093664, Example 6b | (R)-1-(4-(6-amino-5-(tri...)
Affinity DataKd:  0.740nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289481BDBM289481(US10093664, Example 57 | US10093664, Example 62 | ...)
Affinity DataKd:  1.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289491BDBM289491(US10093664, Example 63b | 1-(4-(6-amino-5- (triflu...)
Affinity DataKd:  1.60nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289437BDBM289437(US10093664, Example 18 | 4-(3-(2-cyclopropyl-4-(3-...)
Affinity DataKd:  1.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289489BDBM289489(US10093664, Example 61 | 1-(4-(6-amino-5-(tri- flu...)
Affinity DataKd:  2.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289425BDBM289425(US10093664, Example 5b | (R)-(4-(6-amino-5-(triflu...)
Affinity DataKd:  2.30nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289484BDBM289484(US10093664, Example 60 | (4-(6-amino-5-(trifluoro-...)
Affinity DataKd:  2.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289447BDBM289447(US10093664, Example 28 | 4-(3-(2-isopropyl-4-(1-(1...)
Affinity DataKd:  2.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289466BDBM289466(US10093664, Example 42 | 5-(2-(cyclopropyl- methyl...)
Affinity DataKd:  3.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289509BDBM289509(US10093664, Example 74 | 5-(2-isopropyl-1-(3-(4- m...)
Affinity DataKd:  4.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289480BDBM289480(US10093664, Example 56 | (4-(6-amino-5-(tri- fluor...)
Affinity DataKd:  5.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289471BDBM289471(US10093664, Example 47 | 5-(2-isobutyl-1-(3- morph...)
Affinity DataKd:  6nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289444BDBM289444(US10093664, Example 25 | 5-(1-(3-(bis(2-methoxyeth...)
Affinity DataKd:  6.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289455BDBM289455(US10093664, Example 32 | 5-(1-(3-morpholino- bicyc...)
Affinity DataKd:  6.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289443BDBM289443(US10093664, Example 24 | 5-(2-cyclopropyl-1-(3-((2...)
Affinity DataKd:  6.80nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289436BDBM289436(US10093664, Example 17 | 5-(2-cyclopropyl-1-(3-(4-...)
Affinity DataKd:  6.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289445BDBM289445(US10093664, Example 26 | 1-(3-(4-(6-amino-5-(trifl...)
Affinity DataKd:  7nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289458BDBM289458(US10093664, Example 35 | 5-(2-(cyclopropyl- methyl...)
Affinity DataKd:  7.20nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289511BDBM289511(US10093664, Example 76 | 5-(2-cyclopropyl-1-(3- (4...)
Affinity DataKd:  7.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289510BDBM289510(US10093664, Example 75 | 5-(2-cyclopropyl-1-(3- (4...)
Affinity DataKd:  7.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289424BDBM289424(US10093664, Example 4)
Affinity DataKd:  8.30nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289473BDBM289473(US10093664, Example 49 | US10093664, Example 51 | ...)
Affinity DataKd:  8.60nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289474BDBM289474(US10093664, Example 50 | 5-(2-(sec-butyl)-1-(3- mo...)
Affinity DataKd:  9.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289441BDBM289441(US10093664, Example 22 | 4-(3-(4-(6-amino-5-(trifl...)
Affinity DataKd:  9.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289456BDBM289456(US10093664, Example 33 | (S)-1-(4-(6-amino-5- (tri...)
Affinity DataKd:  9.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289423BDBM289423(US10093664, Example 3 | 5-(2-isopropyl-1-(3-morpho...)
Affinity DataKd:  11nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289478BDBM289478(US10093664, Example 54 | 1-(4-(6-amino-5-(tri- flu...)
Affinity DataKd:  11nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289421BDBM289421(US10093664, Example 1 | 5-(2-cyclopropyl-1-(3-morp...)
Affinity DataKd:  11.4nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289504BDBM289504(US10093664, Example 68 | 1-(4-(6-amino-5-(tri- flu...)
Affinity DataKd:  13nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289506BDBM289506(US10093664, Example 71 | 3-(difluoromethoxy)-5- (1...)
Affinity DataKd:  13nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289472BDBM289472(US10093664, Example 48 | 5-(1-(3-morpholino- bicyc...)
Affinity DataKd:  13nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289422BDBM289422(US10093664, Example 2)
Affinity DataKd:  13nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289479BDBM289479(US10093664, Example 55 | 1-(4-(6-amino-5-(tri- flu...)
Affinity DataKd:  14nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289492BDBM289492(US10093664, Example 64 | 5-(2-((benzyloxy)- methyl...)
Affinity DataKd:  14nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289438BDBM289438(US10093664, Example 19 | 5-(2-cyclopropyl-1-(3-(pi...)
Affinity DataKd:  14nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289430BDBM289430(US10093664, Example 11 | 5-(1-isopropyl-5-(3-morph...)
Affinity DataKd:  15nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289469BDBM289469(US10093664, Example 45 | 5-(2-isobutyl-1-(3- morph...)
Affinity DataKd:  15nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289442BDBM289442(US10093664, Example 23 | 1-(3-(4-(6-amino-5-(trifl...)
Affinity DataKd:  17nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289508BDBM289508(US10093664, Example 73 | 5-(2-(cyclopropyl- methyl...)
Affinity DataKd:  18nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289482BDBM289482(US10093664, Example 58 | (4-(6-amino-5-(trifluoro-...)
Affinity DataKd:  18nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289434BDBM289434(US10093664, Example 15 | 5-(2-cyclopropyl-1-(3-(4-...)
Affinity DataKd:  18nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289460BDBM289460(US10093664, Example 37 | 5-(2-cyclopropyl-1-(3- mo...)
Affinity DataKd:  19nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289461BDBM289461(US10093664, Example 38 | 3-(difluoromethoxy)-5- (2...)
Affinity DataKd:  19nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandChemical structure of BindingDB Monomer ID 289507BDBM289507(US10093664, Example 72 | 5-(2-(cyclopropyl- methyl...)
Affinity DataKd:  19nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

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