Compile Data Set for Download or QSAR
Report error Found 590 Enz. Inhib. hit(s) with all data for entry = 1376
TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319469BDBM319469((3-cyanophenyl) methyl N-{4-[2- ({[(cyclopropyl- c...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319153BDBM319153(US10173991, Example 196 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319472BDBM319472(2,2,2-trifluoroethyl N-{4-[2- ({[(cyclopropyl- ca...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319011BDBM319011(US10173991, Example 52 | benzyl N-{4-[2- ({[(cyclo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319458BDBM319458(2-(6-{4-[(benzyl- carbamoyl) amino]phenyl}- 5-fluo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319525BDBM319525(5-amino-1-{4-[2- ({[(cyclopropyl- carbamoyl)methyl...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319013BDBM319013(US10173991, Example 54 | benzyl N-(4-{2- [cyclohex...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319205BDBM319205(US10173991, Example 248 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319332BDBM319332(US10173991, Example 377 | N-({[2- (benzyloxy)ethyl...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319524BDBM319524(2-{6-[4-(5-amino- 4-cyano-1H- pyrazol-1-yl) phenyl...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319335BDBM319335(US10173991, Example 380 | 2-[6-(6- fluoropyridin- ...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319483BDBM319483(propan-2-yl N-{4- [2-({[(cyclopropyl- carbamoyl)me...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 318970BDBM318970(US10173991, Example 11 | benzyl N-(4-{2- [(cyclopr...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319101BDBM319101(US10173991, Example 144 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319474BDBM319474(cyclopropylmethyl N-{4-[2- [(cyclopropyl- carbamo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319477BDBM319477(cyclopropylmethyl N-{4-[2- ({[(cyclopropyl- carba...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 318967BDBM318967(US10173991, Example 8 | benzyl N-{4-[2- ({[(cyclop...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319094BDBM319094(US10173991, Example 137 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 318969BDBM318969(US10173991, Example 10 | benzyl N-{4-[2- ({[(cyclo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 318968BDBM318968(US10173991, Example 9 | benzyl N-{4-[2- ({[(cyclop...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319499BDBM319499(benzyl N-(3-{2- [(cyclopropane- sulfonyl) ({[(cycl...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319050BDBM319050(US10173991, Example 93 | N-[(cyclopropyl- carbamoy...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319375BDBM319375(benzyl N-{4-[2- ({[(cyclopropyl- carbamoyl)methyl]...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319495BDBM319495(benzyl N-{5-[2- ({[(cyclopropyl- carbamoyl)methyl]...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319494BDBM319494(benzyl N-{3-[2- ({[(cyclopropyl- carbamoyl)methyl]...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319497BDBM319497(benzyl N-{3-[2- ({[(cyclopropyl- carbamoyl)methyl]...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319496BDBM319496(benzyl N-{5-[2- ({[(cyclopropyl- carbamoyl)methyl]...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319515BDBM319515(4-[2- ({[(cyclopropyl- carbamoyl)methyl] carbamoyl...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319517BDBM319517(N-{4-[2- ({[(cyclopropyl- carbamoyl)methyl] carbam...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319516BDBM319516(N-{4-[2- ({[(cyclopropyl- carbamoyl)methyl] carbam...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319007BDBM319007(US10173991, Example 48 | benzyl N-{4-[2- ({[(cyclo...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319442BDBM319442(N-[(cyclopropyl- carbamoyl) methyl]-2- (dimethyl- ...)
Affinity DataIC50: 1nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319467BDBM319467(pyridin-2- ylmethyl N-{4-[2- ({[(cyclopropyl- carb...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319466BDBM319466(pyridin-2- ylmethyl N-{4-[2- ({[(cyclopropyl- carb...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319082BDBM319082(US10173991, Example 125 | methyl N-{4-[4- chloro-2...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319533BDBM319533(2-[6-(2- cyclopropyl- 1-oxo-2,3-dihydro- 1H-isoind...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319331BDBM319331(US10173991, Example 375 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319012BDBM319012(US10173991, Example 53 | benzyl N-(4-{2- [(butane-...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319081BDBM319081(US10173991, Example 124 | methyl N-{4-[4- chloro-2...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319098BDBM319098(US10173991, Example 141 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319485BDBM319485(propan-2-yl N-{4- [2-({[(cyclopropyl- carbamoyl)me...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319484BDBM319484(propan-2-yl N-{4- [2-({[(cyclopropyl- carbamoyl)me...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319486BDBM319486(propan-2-yl N-(4- {2-[(cyclopropane- sulfonyl) ({[...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319105BDBM319105(US10173991, Example 148 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319475BDBM319475(2,2,2-trifluoroethyl N-{4-[2- ({[(cyclopropyl- ca...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319091BDBM319091(US10173991, Example 134 | tert-butyl 3-[2- ({[(cyc...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319479BDBM319479(2-methoxyethyl N-{4-[2- ({[(cyclopropyl- carbamoy...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319481BDBM319481(2-methoxyethyl N-(4-{2- [(cyclopropane- sulfonyl)...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319161BDBM319161(US10173991, Example 204 | N-[(cyclopropyl- carbamo...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEndothelial lipase(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 319544BDBM319544(N-[(cyclopropyl- carbamoyl) methyl]-2-(5- fluoro-6...)
Affinity DataIC50: 2nMAssay Description:Endothelial lipase (EL) and hepatic lipase (HL) activities were measured using a fluorescent substrate, A10070, (Invitrogen, CA) doped into an artifi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

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