Compile Data Set for Download or QSAR
Report error Found 296 Enz. Inhib. hit(s) with all data for entry = 9512
TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472033BDBM472033(US10829480, Example SC_2061)
Affinity DataKi:  0.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472009BDBM472009(US10829480, Example SC_2019 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  0.800nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471982BDBM471982(US10829480, Example SC_2006 | CIS-2-[[1-(Cyclobuty...)
Affinity DataKi:  0.800nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472098BDBM472098(US10829480, Example SC_2093 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  0.800nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471984BDBM471984(US10829480, Example SC_2007 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  1.10nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472075BDBM472075(US10829480, Example SC_2081 | CIS-3-[[1-(Cyclobuty...)
Affinity DataKi:  1.20nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472105BDBM472105(US10829480, Example SC_2096 | CIS-3-Benzy1-1-(cycl...)
Affinity DataKi:  1.30nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472053BDBM472053(US10829480, Example SC_2103 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  1.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472091BDBM472091(US10829480, Example SC_2089 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  1.80nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472089BDBM472089(US10829480, Example SC_2088 | CIS-3-[[1-(Cyclobuty...)
Affinity DataKi:  1.90nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472120BDBM472120(US10829480, Example SC_2159 | CIS-2-[4-[[1-(Cyclob...)
Affinity DataKi:  2.35nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472058BDBM472058(US10829480, Example SC_2105 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  2.40nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471850BDBM471850(US10829480, Example SC_2001 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  2.70nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471985BDBM471985(US10829480, Example SC_2039 | CIS-1-(3,3-Difluoro-...)
Affinity DataKi:  2.80nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472044BDBM472044(US10829480, Example SC_2036 | CIS-8-Dimethylamino-...)
Affinity DataKi:  3.10nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472051BDBM472051(US10829480, Example SC_2102 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  3.30nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472059BDBM472059(US10829480, Example SC_2074 | CIS-1-[[8-Dimethylam...)
Affinity DataKi:  3.40nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472097BDBM472097(US10829480, Example SC_2125 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  3.40nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472085BDBM472085(US10829480, Example SC_2086 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  3.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472017BDBM472017(US10829480, Example SC_2023 | CIS-1-(Cyclopentyl-m...)
Affinity DataKi:  3.80nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472083BDBM472083(US10829480, Example SC_2085 | CIS-4-[[1-(Cyclobuty...)
Affinity DataKi:  3.80nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472095BDBM472095(US10829480, Example SC_2124 | CIS-8-Dimethylamino-...)
Affinity DataKi:  4nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472076BDBM472076(US10829480, Example SC_2113 | CIS-8-Dimethylamino-...)
Affinity DataKi:  4nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472121BDBM472121(US10829480, Example SC_2160 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  4nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471883BDBM471883(US10829480, Example SC_2002 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  4.30nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472034BDBM472034(US10829480, Example SC_2031 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  4.60nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472015BDBM472015(US10829480, Example SC_2022 | CIS-8-Dimethylamino-...)
Affinity DataKi:  5.40nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472096BDBM472096(US10829480, Example SC_2092 | CIS-2-[[1-(Cyclobuty...)
Affinity DataKi:  5.60nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472001BDBM472001(CIS-1-Butyl-8-dimethylamino-3-[(4-methoxyphenyl)-m...)
Affinity DataKi:  6.40nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472139BDBM472139(US10829480, Example SC_2174 | CIS-8-Dimethylamino-...)
Affinity DataKi:  8.15nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472012BDBM472012(US10829480, Example SC_2051 | CIS-8-Dimethylamino-...)
Affinity DataKi:  9nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472061BDBM472061(US10829480, Example SC_2075 | CIS-8-Dimethylamino-...)
Affinity DataKi:  9.10nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472065BDBM472065(US10829480, Example SC_2108 | CIS-8-Dimethylamino-...)
Affinity DataKi:  10.1nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471997BDBM471997(CIS-1-(Cyclobutyl-methyl)-3-[(4-methoxyphenyl)-met...)
Affinity DataKi:  10.8nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472024BDBM472024(US10829480, Example SC_2026 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  11nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472102BDBM472102(US10829480, Example SC_2095 | CIS-8-Dimethylamino-...)
Affinity DataKi:  11.2nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472010BDBM472010(US10829480, Example SC_2050 | CIS-8-Dimethylamino-...)
Affinity DataKi:  11.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472047BDBM472047(US10829480, Example SC_2100 | CIS-3-[8-Dimethylami...)
Affinity DataKi:  11.8nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472027BDBM472027(US10829480, Example SC_2027 | CIS-3-[[1-(Cyclobuty...)
Affinity DataKi:  12nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472117BDBM472117(US10829480, Example SC_2155 | CIS-2-[4-[[8-Dimethy...)
Affinity DataKi:  12.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472124BDBM472124(US10829480, Example SC_2163 | CIS-2-[4-[[1-(Cyclob...)
Affinity DataKi:  13nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471983BDBM471983(US10829480, Example SC_2038 | CIS-1-(2-Cyclobutyl-...)
Affinity DataKi:  13.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472048BDBM472048(US10829480, Example SC_2069 | CIS-8-Dimethylamino-...)
Affinity DataKi:  14nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472011BDBM472011(US10829480, Example SC_2020 | CIS-1-(Cyclobutyl-me...)
Affinity DataKi:  15.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472060BDBM472060(US10829480, Example SC_2106 | CIS-3-[[1-[(5-Cyano-...)
Affinity DataKi:  16.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472069BDBM472069(US10829480, Example SC_2110 | CIS-3-[[8-Dimethylam...)
Affinity DataKi:  16.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471992BDBM471992(CIS-2-[8-Dimethylamino-3-[(4-methoxyphenyl)-methyl...)
Affinity DataKi:  16.5nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472067BDBM472067(US10829480, Example SC_2109 | CIS-2-[[8-Dimethylam...)
Affinity DataKi:  17nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 471989BDBM471989(CIS-4-[[1-(Cyclobutyl-methyl)-8-dimethylamino-2-ox...)
Affinity DataKi:  17.6nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Gruenenthal

US Patent
LigandChemical structure of BindingDB Monomer ID 472037BDBM472037(US10829480, Example SC_2063 | CIS-2-[8-Dimethylami...)
Affinity DataKi:  18nMAssay Description:Mu-Opioid Peptide (hMOP): The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

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