Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 9791
LigandChemical structure of BindingDB Monomer ID 489224BDBM489224(US10961233, Example 85)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489223BDBM489223(US10961233, Example 84)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489222BDBM489222(US10961233, Example 77)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489221BDBM489221(US10961233, Example 76)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489220BDBM489220(US10961233, Example 75)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489218BDBM489218(US10961233, Example 74)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489216BDBM489216(US10961233, Example 72)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489215BDBM489215(US10961233, Example 70)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489214BDBM489214(US10961233, Example 69)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 489212BDBM489212(US10961233, Example 67)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489209BDBM489209(US10961233, Example 64)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489208BDBM489208(US10961233, Example 63)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489200BDBM489200(US10961233, Example 55)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489199BDBM489199(US10961233, Example 54)
Affinity DataIC50: 10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489196BDBM489196(US10961233, Example 45)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489195BDBM489195(US10961233, Example 44)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489226BDBM489226(US10961233, Example 87)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489225BDBM489225(US10961233, Example 86)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489187BDBM489187(US10961233, Example 28)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489186BDBM489186(US10961233, Example 25)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489185BDBM489185(US10961233, Example 24)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489217BDBM489217(US10961233, Example 73)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489184BDBM489184(US10961233, Example 23)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489182BDBM489182(US10961233, Example 21)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 488654BDBM488654(US10961233, Example 20)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489213BDBM489213(US10961233, Example 68)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489211BDBM489211(US10961233, Example 66)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489210BDBM489210(US10961233, Example 65)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489207BDBM489207(US10961233, Example 62)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489206BDBM489206(US10961233, Example 61)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489205BDBM489205(US10961233, Example 60)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489204BDBM489204(US10961233, Example 59)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489202BDBM489202(US10961233, Example 57)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489201BDBM489201(US10961233, Example 56)
Affinity DataIC50: 17.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489194BDBM489194(US10961233, Example 35)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489193BDBM489193(US10961233, Example 34)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489192BDBM489192(US10961233, Example 33)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489191BDBM489191(US10961233, Example 32)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489190BDBM489190(US10961233, Example 31)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489188BDBM489188(US10961233, Example 29)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489203BDBM489203(US10961233, Example 58)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489198BDBM489198(US10961233, Example 53)
Affinity DataIC50: 62.5nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 488641BDBM488641(US10961233, Example 19 | US10961233, Example 22)
Affinity DataIC50: 100nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489189BDBM489189(US10961233, Example 30)
Affinity DataIC50: 100nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 488641BDBM488641(US10961233, Example 19 | US10961233, Example 22)
Affinity DataIC50: 100nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 489197BDBM489197(US10961233, Example 46)
Affinity DataIC50: 100nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
US Patent