Compile Data Set for Download or QSAR
Report error Found 291 Enz. Inhib. hit(s) with all data for entry = 10511
LigandChemical structure of BindingDB Monomer ID 542862BDBM542862(4-(3-((2-(4-(difluoromethoxy)phenyl)-8-methoxy-2,3...)
Affinity DataIC50: 2nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542881BDBM542881(3-((2-(6-ethoxypyridin-3-yl)-8-methoxy-2,3-dihydro...)
Affinity DataIC50: 2nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542814BDBM542814(4-(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dih...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542815BDBM542815(6-methoxy-3-((8-methoxy-2-(6-methoxypyridin-3-yl)-...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542847BDBM542847(3-((2-(6-ethylpyridin-3-yl)-8-methoxy-2,3-dihydrob...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542975BDBM542975(3-(3-methoxy-4-((6-methoxypyridin-3-yl)methoxy)ben...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542818BDBM542818(4-(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dih...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542819BDBM542819(4-(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dih...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542824BDBM542824(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542551BDBM542551(US11274108, Example 1-4 | 3-((2-(4-methoxyphenyl)-...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542813BDBM542813(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542721BDBM542721(US11274108, Example 1-23 | 4-(3-((2-(6-methoxypyri...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542791BDBM542791((S)-6-(difluoromethyl)-3-((8-methoxy-2-(6-methoxyp...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542519BDBM542519(US11274108, Example 1-2-enant-B | (S)-4-(3-((2-(4-...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542518BDBM542518(US11274108, Example 1-2-enant-A | (S)-4-(3-((2-(4-...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542974BDBM542974(3-(3-methoxy-4-((6-methoxypyridin-3-yl)methoxy)ben...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542816BDBM542816(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542848BDBM542848(3-((2-(6-ethylpyridin-3-yl)-8-methoxy-2,3-dihydrob...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542753BDBM542753(US11274108, Example 1-53 | 3-((8-methoxy-2-(6-meth...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542820BDBM542820(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542516BDBM542516(US11274108, Example 1-1 | 4-(1-((2-(4-methoxypheny...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542777BDBM542777(US11274108, Example 1-75 | 6-(1,3-dimethyl-1H-pyra...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542553BDBM542553(US11274108, Example 1-5-enant-A | (S)-4-(3-((2-(6-...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542851BDBM542851(4-(3-((8-methoxy-2-(4-methoxyphenyl)-2,3-dihydrobe...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542688BDBM542688(US11274108, Example 1-12 | 4-(3-((2-(4-methoxyphen...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542517BDBM542517(US11274108, Example 1-2 | 4-(3-((2-(4-methoxypheny...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542759BDBM542759(US11274108, Example 1-59 | 4-(3-((8-methoxy-2-(6-m...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542811BDBM542811(6-bromo-3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542944BDBM542944(7-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542879BDBM542879(3-((2-(6-ethoxypyridin-3-yl)-8-methoxy-2,3-dihydro...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542727BDBM542727(US11274108, Example 1-29 | 4-(3-((8-fluoro-2-(4-(t...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542855BDBM542855(4-(3-((2-(4-(difluoromethoxy)phenyl)-8-methoxy-2,3...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542831BDBM542831(3-((2-(6-cyclopropylpyridin-3-yl)-8-methoxy-2,3-di...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542770BDBM542770(US11274108, Example 1-68 | 3-((8-methoxy-2-(6-meth...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542852BDBM542852(3-((8-methoxy-2-(4-methoxyphenyl)-2,3-dihydrobenzo...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542771BDBM542771(US11274108, Example 1-69 | 6-(1H-imidazol-1-yl)-3-...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542761BDBM542761(US11274108, Example 1-60-enant-A | 6-methoxy-3-((8...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542754BDBM542754(US11274108, Example 1-54 | 4-(3-((8-methoxy-2-(6-m...)
Affinity DataIC50: 9nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542778BDBM542778(US11274108, Example 1-76 | 6-(6-fluoropyridin-3-yl...)
Affinity DataIC50: 9nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542841BDBM542841(3-((8-methoxy-2-(6-methylpyridin-3-yl)-2,3-dihydro...)
Affinity DataIC50: 9nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542750BDBM542750(US11274108, Example 1-52 | 4-(3-((8-methoxy-2-(6-m...)
Affinity DataIC50: 10nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542860BDBM542860(3-((2-(4-(difluoromethoxy)phenyl)-8-methoxy-2,3-di...)
Affinity DataIC50: 10nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542846BDBM542846(3-((2-(6-ethylpyridin-3-yl)-8-methoxy-2,3-dihydrob...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542751BDBM542751(US11274108, Example 1-52-enant-A | 4-(3-((8-methox...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542786BDBM542786(US11274108, Example 1-83-enant-A | azetidin-1-yl(3...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542825BDBM542825(3-((2-(6-cyclopropylpyridin-3-yl)-8-methoxy-2,3-di...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542827BDBM542827(3-((2-(6-cyclopropylpyridin-3-yl)-8-methoxy-2,3-di...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542738BDBM542738(US11274108, Example 1-40 | 3-((8-fluoro-2-(6-metho...)
Affinity DataIC50: 12nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542737BDBM542737(US11274108, Example 1-39 | 4-(3-((8-fluoro-2-(6-me...)
Affinity DataIC50: 12nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542760BDBM542760(US11274108, Example 1-60 | 6-methoxy-3-((8-methoxy...)
Affinity DataIC50: 12nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

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