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Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 7387
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192505BDBM192505(US9187477, 1)
Affinity DataEC50:  1.20nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192510BDBM192510(US9187477, 6)
Affinity DataEC50:  6nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192508BDBM192508(US9187477, 16 | US9187477, 4)
Affinity DataEC50:  12nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192513BDBM192513(US9187477, 9)
Affinity DataEC50:  17nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192514BDBM192514(US9187477, 10)
Affinity DataEC50:  26nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192506BDBM192506(US9187477, 2)
Affinity DataEC50:  32nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192515BDBM192515(US9187477, 11)
Affinity DataEC50:  35nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192507BDBM192507(US9187477, 3)
Affinity DataEC50:  108nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192509BDBM192509(US9187477, 5)
Affinity DataEC50:  119nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192519BDBM192519(US9187477, 15)
Affinity DataEC50:  133nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192508BDBM192508(US9187477, 16 | US9187477, 4)
Affinity DataEC50:  290nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192512BDBM192512(US9187477, 8)
Affinity DataEC50:  339nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192511BDBM192511(US9187477, 7)
Affinity DataEC50:  468nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192518BDBM192518(US9187477, 14)
Affinity DataEC50:  578nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192516BDBM192516(US9187477, 12)
Affinity DataEC50:  1.31E+3nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 192517BDBM192517(US9187477, 13)
Affinity DataEC50:  2.04E+3nMpH: 7.0Assay Description:In the 384-well plates 1.25 ul of test compound in assay buffer (20 mM HEPES pH 7.0, 0.025% BSA, 15 mM MgCl2, 0.01% Brij) was mixed with 1.25 ul of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent