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TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50200169(6-methyl-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl...)
Affinity DataKi:  0.0370nMAssay Description:Displacement of [3H]CP-55,940 from CB2 receptor in CD-1 mouse spleen homogenate after 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM21280(N-(1,3,3-trimethylbicyclo(2.2.1)heptan-2-yl)-5-(4-...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2012
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50200169(6-methyl-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM21280(N-(1,3,3-trimethylbicyclo(2.2.1)heptan-2-yl)-5-(4-...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2012
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50532777(CHEMBL4470925)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50233601(CHEMBL4062745)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50463772(CHEMBL4239190)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]CP-55,940 from recombinant mouse Cb2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50532777(CHEMBL4470925)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50532778(CHEMBL4465566 | US10882838, Example 3.6)
Affinity DataKi:  0.200nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3-(1,1-dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50532778(CHEMBL4465566 | US10882838, Example 3.6)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3-(1,1-dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50532778(CHEMBL4465566 | US10882838, Example 3.6)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50130624((6aR,10aR)-3-(2-hexyl-1,3-dioxolan-2-yl)-6,6,9-tri...)
Affinity DataKi:  0.220nMAssay Description:Compound was tested for its binding affinity against mouse spleen Cannabinoid receptor 2 using [3H]CP-55940 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]-CP-55940 from cannabinoid CB2 receptor in CD1 mouse spleen membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50121425((6aR,10aR)-3-(2,2-Dichloro-1-hexyl-cyclopropyl)-6,...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity for Cannabinoid receptor 2 by the ability to displace radiolabeled CP-55940 from mouse spleen synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50176977(1,4-dihydroindeno[1,2-c]-pyrazole | 6-chloro-1-(2'...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]CP-55940 from CD1 mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50176977(1,4-dihydroindeno[1,2-c]-pyrazole | 6-chloro-1-(2'...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in CD1 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50080030(3-Heptyl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity towards Cannabinoid receptor 2 in mouse spleen membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM21244(CP-56667 [(+)-AC],XV | CP-55,940 | 2-[(1S,2S,5S)-5...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at mouse CB2 receptor transfected in CHO-K1 cells assessed as beta2-arrestin recruitment incubated for 90 mins by luminescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50176979(8-methyl-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in CD1 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50067735((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  0.490nMAssay Description:Compound was tested for its binding affinity against mouse spleen Cannabinoid receptor 2 using [3H]CP-55940 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50067735((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity for Cannabinoid receptor 2 by the ability to displace radiolabeled CP-55940 from mouse spleen synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM474533(US10882838, Example 1.5)
Affinity DataKi:  0.5nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50233622(CHEMBL4073011 | US10882838, Example 1.35)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM474531(US10882838, Example 1.3)
Affinity DataKi:  0.5nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50233622(CHEMBL4073011 | US10882838, Example 1.35)
Affinity DataKi:  0.5nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50463775(CHEMBL4240671)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CP-55,940 from recombinant mouse Cb2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50063885((6aR,10aR)-3-(2-Hexyl-[1,3]dithiolan-2-yl)-6,6,9-t...)
Affinity DataKi:  0.520nMAssay Description:Compound was tested for its binding affinity against mouse spleen Cannabinoid receptor 2 using [3H]CP-55940 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50063885((6aR,10aR)-3-(2-Hexyl-[1,3]dithiolan-2-yl)-6,6,9-t...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity for Cannabinoid receptor 2 by the ability to displace radiolabeled CP-55940 from mouse spleen synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50063885((6aR,10aR)-3-(2-Hexyl-[1,3]dithiolan-2-yl)-6,6,9-t...)
Affinity DataKi:  0.520nMAssay Description:The compound was evaluated for its affinity towards cannabinoid receptor 2 (CB2) in mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2012
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM474532(US10882838, Example 1.4)
Affinity DataKi:  0.600nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM474530(US10882838, Example 1.2)
Affinity DataKi:  0.600nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50111517(CHEMBL3605054)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor in mouse spleen membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50176976(8-chloro-1-(2',4'-dichlorophenyl)-N-cyclohexyl-1,4...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in CD1 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50233605(CHEMBL3104362 | US10882838, Example 1.20)
Affinity DataKi:  0.700nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50557516(CHEMBL4787347)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM474537(US10882838, Example 1.9)
Affinity DataKi:  0.700nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50213889(3-[(Z)-5,6,7,8-tetrahydro-naphthalen-1-ylimino]-2-...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50233602(CHEMBL4071389 | US10882838, Example 1.8)
Affinity DataKi:  0.700nMAssay Description:All the cannabinoids discussed in this invention are tested for their ability to bind to CB1 and CB2 receptors using membranes from rat brain or HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
US Patent

TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50330773(JWH-051 | CHEMBL1277685 | ((6aR,10aR)-6,6-dimethyl...)
Affinity DataKi:  0.720nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2012
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM21244(CP-56667 [(+)-AC],XV | CP-55,940 | 2-[(1S,2S,5S)-5...)
Affinity DataKi:  0.730nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2012
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50582401(CHEMBL5081770)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50582400(CHEMBL5077315)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50582403(CHEMBL5085420)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50233602(CHEMBL4071389 | US10882838, Example 1.8)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50233606(CHEMBL4068675)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50582406(CHEMBL5091754)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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