Compile Data Set for Download or QSAR
Report error Found 127 of affinity data for UniProtKB/TrEMBL: Q03405
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402366(CHEMBL2206696)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50005398(CHEMBL2206694)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402361(CHEMBL2206680)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402378(CHEMBL2206685)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402373(CHEMBL2206691)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402360(CHEMBL2206681)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402372(CHEMBL2206692)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402371(CHEMBL2206693)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402374(CHEMBL2206690)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402362(CHEMBL2206700)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402363(CHEMBL2206699)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402375(CHEMBL2206689)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402370(CHEMBL2206683)
Affinity DataKi:  0.00600nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402367(CHEMBL2206695)
Affinity DataKi:  0.00700nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402376(CHEMBL2206688)
Affinity DataKi:  0.00800nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402364(CHEMBL2206698)
Affinity DataKi:  0.0110nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402365(CHEMBL2206697)
Affinity DataKi:  0.0120nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402377(CHEMBL2206687)
Affinity DataKi:  0.0330nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402379(CHEMBL2206686)
Affinity DataKi:  0.296nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402368(CHEMBL2206682)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402369(CHEMBL1652555)
Affinity DataKi:  20.8nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120747(cyclic uPA-derived peptide | CHEMBL412236)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120746(cyclic uPA-derived peptide | CHEMBL405302)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120740(cyclic uPA-derived peptide | CHEMBL405999)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120745(cyclic uPA-derived peptide | CHEMBL263158)
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120743(cyclic uPA-derived peptide | CHEMBL385968)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222392(IPR-2260 (45))
Affinity DataKi:  400nM IC50: 1.57E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50549787(CHEMBL4791246)
Affinity DataIC50: 500nMAssay Description:Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50549794(CHEMBL4753144)
Affinity DataIC50: 500nMAssay Description:Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222393(IPR-1609 (46))
Affinity DataKi:  600nM IC50: 2.16E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222350(IPR-1110 (1))
Affinity DataKi:  700nM IC50: 1.84E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120749(cyclic uPA-derived peptide | CHEMBL412223)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222391(IPR-1607 (44))
Affinity DataKi:  800nM IC50: 2.40E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222386(IPR-1168 (39))
Affinity DataKi:  900nM IC50: 2.31E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120742(cyclic uPA-derived peptide | CHEMBL264653)
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222351(IPR-1201 (4))
Affinity DataKi:  1.00E+3nM IC50: 1.63E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222354(IPR-1178 (7))
Affinity DataKi:  1.10E+3nM IC50: 2.02E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222370(IPR-1174 (23))
Affinity DataKi:  1.20E+3nM IC50: 1.84E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222364(IPR-1182 (17))
Affinity DataKi:  1.30E+3nM IC50: 3.71E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222360(IPR-1171 (13))
Affinity DataKi:  1.30E+3nM IC50: 2.30E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222362(IPR-1195 (15))
Affinity DataKi:  1.60E+3nM IC50: 6.17E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222356(IPR-1185 (9))
Affinity DataKi:  1.70E+3nM IC50: 3.56E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222358(IPR-1193 (11))
Affinity DataKi:  1.70E+3nM IC50: 5.78E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222369(IPR-1176 (22))
Affinity DataKi:  1.90E+3nM IC50: 5.38E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222383(IPR-1160 (36))
Affinity DataKi:  1.90E+3nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222357(IPR-1192 (10))
Affinity DataKi:  1.90E+3nM IC50: 3.01E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222373(IPR-1188 (26))
Affinity DataKi:  2.00E+3nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222359(IPR-1175 (12))
Affinity DataKi:  2.00E+3nM IC50: 4.52E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222376(IPR-1191 (29))
Affinity DataKi:  2.10E+3nM IC50: 2.95E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM222363(IPR-1186 (16))
Affinity DataKi:  2.10E+3nM IC50: 3.53E+4nMAssay Description:Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2017
Entry Details Article
PubMed
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