Compile Data Set for Download or QSAR
Report error Found 17 of affinity data for UniProtKB/TrEMBL: Q499N1
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133122BDBM50133122(5-[2'-(2,2-Difluoro-ethoxy)-3',5'-diisopropyl-biph...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032671BDBM50032671(6-[1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-nap...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133126BDBM50133126(5-[2-(3,5-Diisopropyl-2-propoxy-phenyl)-cyclopent-...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133114BDBM50133114(5-{2-[2-(3-Fluoro-propoxy)-3,5-diisopropyl-phenyl]...)
Affinity DataKi:  2.48E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133118BDBM50133118(5-{3-[2-(2,2-Difluoro-ethoxy)-3,5-diisopropyl-phen...)
Affinity DataKi:  2.57E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129720BDBM50129720(7-[3,5-Di-tert-butyl-2-(2,2-difluoro-ethoxy)-pheny...)
Affinity DataKi:  2.75E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133127BDBM50133127(5-{3-[2-(3-Fluoro-propoxy)-3,5-diisopropyl-phenyl]...)
Affinity DataKi:  3.41E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133120BDBM50133120(5-{3-[3,5-Diisopropyl-2-(2,2,2-trifluoro-ethoxy)-p...)
Affinity DataKi:  3.44E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133117BDBM50133117(5-{2-[2-(3-Fluoro-propoxy)-3,5-diisopropyl-phenyl]...)
Affinity DataKi:  3.67E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133128BDBM50133128(5-{2-[2-(2,2-Difluoro-ethoxy)-3,5-diisopropyl-phen...)
Affinity DataKi:  3.73E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133116BDBM50133116((2E,4E)-5-{3-[3,5-Di-tert-butyl-2-(3,3-difluoro-pr...)
Affinity DataKi:  5.41E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133121BDBM50133121(5-{3-[3-tert-Butyl-2-(2,2-difluoro-ethoxy)-5-ethyl...)
Affinity DataKi:  5.65E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133115BDBM50133115(5-[2'-(3-Fluoro-propoxy)-3',5'-diisopropyl-bipheny...)
Affinity DataKi:  7.50E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133119BDBM50133119(5-{2-[3,5-Diisopropyl-2-(2,2,2-trifluoro-ethoxy)-p...)
Affinity DataKi:  8.79E+3nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133125BDBM50133125(5-{3-[3,5-Diisopropyl-2-(2,2,2-trifluoro-ethoxy)-p...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133124BDBM50133124(5-[3',5'-Di-tert-butyl-2'-(3-fluoro-propoxy)-biphe...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor, alpha, isoform CRA_b(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133123BDBM50133123(5-{3-[3-tert-Butyl-5-ethyl-2-(3-fluoro-propoxy)-ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for Retinoic acid receptor alpha was determined by competing with 3[H]-ATRAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed