Compile Data Set for Download or QSAR
Report error Found 716 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 5A'
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148155BDBM148155(US8962612, 26)
Affinity DataKi:  0.680nM ΔG°:  -54.4kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148163BDBM148163(US8962612, 66)
Affinity DataKi:  0.75nM ΔG°:  -54.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50098551BDBM50098551((R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolid...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity to 5HT5A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148169BDBM148169(US8962612, 80)
Affinity DataKi:  0.850nM ΔG°:  -53.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148165BDBM148165(US8962612, 74)
Affinity DataKi:  0.880nM ΔG°:  -53.8kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148171BDBM148171(US8962612, 86)
Affinity DataKi:  0.950nM ΔG°:  -53.6kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 78940BDBM78940(methanesulfonic acid;1-methyl-4-(3-methylsulfanyl-...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 78940BDBM78940(methanesulfonic acid;1-methyl-4-(3-methylsulfanyl-...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 5A receptor was evaluated using [3H]-5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50175465BDBM50175465(7-methyl-3-[2-(4-quinolin-4-yl-piperazin-1-yl)-eth...)
Affinity DataKi: >1nMAssay Description:Inhibitory activity against 5HT5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50323040BDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148156BDBM148156(US8962612, 28)
Affinity DataKi:  1.10nM ΔG°:  -53.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148154BDBM148154(US8962612, 23)
Affinity DataKi:  1.10nM ΔG°:  -53.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135790BDBM135790(US8853242, 162)
Affinity DataKi:  1.20nM ΔG°:  -50.9kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371998BDBM50371998(CHEMBL404372)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135785BDBM135785(US8853242, 152)
Affinity DataKi:  1.30nM ΔG°:  -50.7kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148167BDBM148167(US8962612, 78)
Affinity DataKi:  1.30nM ΔG°:  -52.8kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135780BDBM135780(US8853242, 60)
Affinity DataKi:  1.30nM ΔG°:  -50.7kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135783BDBM135783(US8853242, 148)
Affinity DataKi:  1.40nM ΔG°:  -50.5kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50585913BDBM50585913(CHEMBL5093295)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50371998BDBM50371998(CHEMBL404372)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135782BDBM135782(US8853242, 147)
Affinity DataKi:  1.60nM ΔG°:  -50.2kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148164BDBM148164(US8962612, 69)
Affinity DataKi:  1.60nM ΔG°:  -52.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50371981BDBM50371981(CHEMBL256694)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135795BDBM135795(US8853242, 192)
Affinity DataKi:  1.80nM ΔG°:  -49.9kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148162BDBM148162(US8962612, 62)
Affinity DataKi:  1.90nM ΔG°:  -51.8kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135792BDBM135792(US8853242, 170)
Affinity DataKi:  1.90nM ΔG°:  -49.8kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Mouse)
University of Alberta

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50130269BDBM50130269(LSD,2-Bromo | (6aR,9R)-5-Bromo-7-methyl-4,6,6a,7,8...)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Mouse)
University of Alberta

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50130269BDBM50130269(LSD,2-Bromo | (6aR,9R)-5-Bromo-7-methyl-4,6,6a,7,8...)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2011
Entry Details
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50371464BDBM50371464(CHEMBL273170)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Mouse)
University of Alberta

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50130269BDBM50130269(LSD,2-Bromo | (6aR,9R)-5-Bromo-7-methyl-4,6,6a,7,8...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards mouse 5-hydroxytryptamine 5A receptor was evaluated using [125I]-2-iodo LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135796BDBM135796(US8853242, 211)
Affinity DataKi:  2.30nM ΔG°:  -49.3kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50585914BDBM50585914(CHEMBL5079273)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148161BDBM148161(US8962612, 61)
Affinity DataKi:  2.5nM ΔG°:  -51.1kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50051944BDBM50051944(3-((1R,2S)-2-Dipropylamino-cyclopropyl)-phenol | C...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148157BDBM148157(US8962612, 44)
Affinity DataKi:  2.70nM ΔG°:  -50.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148166BDBM148166(US8962612, 76)
Affinity DataKi:  2.70nM ΔG°:  -50.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371996BDBM50371996(CHEMBL541993)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50130266BDBM50130266(8-Piperazin-1-yl-naphthalen-2-ol | CHEMBL24462)
Affinity DataKi:  3nMAssay Description:Binding affinity for rodent 5-hydroxytryptamine 5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50056445BDBM50056445(lisuride, (S) | lisuride | N'-((8alpha)-9,10-Dideh...)
Affinity DataKi:  3.10nMAssay Description:Table S2 shows raw Ki data for the current study combined with data collected from the literature for the ten additional compounds.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50585912BDBM50585912(CHEMBL5075486)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135788BDBM135788(US8853242, 160)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135789BDBM135789(US8853242, 161)
Affinity DataKi:  3.40nM ΔG°:  -48.3kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148153BDBM148153(US8962612, 8)
Affinity DataKi:  3.60nM ΔG°:  -50.1kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 135781BDBM135781(US8853242, 114)
Affinity DataKi:  3.70nM ΔG°:  -48.1kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148168BDBM148168(US8962612, 79)
Affinity DataKi:  3.70nM ΔG°:  -50.1kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 148160BDBM148160(US8962612, 60)
Affinity DataKi:  3.90nM ΔG°:  -49.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

Target5-hydroxytryptamine receptor 5A(Mouse)
University of Alberta

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50027065BDBM50027065(12'-hydroxy-2'-methyl-5'alpha-(phenylmethyl)ergota...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2011
Entry Details
PubMed
Target5-hydroxytryptamine receptor 5A(Mouse)
University of Alberta

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50027065BDBM50027065(12'-hydroxy-2'-methyl-5'alpha-(phenylmethyl)ergota...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 5A(Mouse)
University of Alberta

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50027065BDBM50027065(12'-hydroxy-2'-methyl-5'alpha-(phenylmethyl)ergota...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
Astellas Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50585909BDBM50585909(CHEMBL5089996)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
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