Compile Data Set for Download or QSAR
Report error Found 217 Enz. Inhib. hit(s) with Target = 'Transcription initiation factor TFIID subunit 1 [1381-1497]'
LigandChemical structure of BindingDB Monomer ID 346517BDBM346517(o-tolylmethyl 4-(3-hydroxy-3-methyl-but-1-ynyl)-2,...)
Affinity DataIC50: 85nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346549BDBM346549(cyclohexylmethyl 4-(3-hydroxy-3-methyl-but-1-ynyl)...)
Affinity DataIC50: 85.3nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346546BDBM346546(2,2-dimethylpropyl 4-(3-hydroxy-3-methyl-but-1-yny...)
Affinity DataIC50: 93.6nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346501BDBM346501(8-quinolylmethyl 4-(3-cyclopropyl-3-hydroxy-but-1-...)
Affinity DataIC50: 93.9nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346544BDBM346544(cyclopentylmethyl 4-(3-hydroxy-3-methyl-but-1-ynyl...)
Affinity DataIC50: 96.8nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346545BDBM346545(2-methylbutyl 4-(3-hydroxy-3-methyl-but-1-ynyl)-2,...)
Affinity DataIC50: 101nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346512BDBM346512([2-(trifluoromethyl)phenyl]methyl4-(3-hydroxy-3-me...)
Affinity DataIC50: 105nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346492BDBM346492(US10202378, Example 98a | US10202378, Example 98b ...)
Affinity DataIC50: 108nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346554BDBM346554(isobutyl 4-[(3R)-3-hydroxy-3-(5-methylisoxazol-3-y...)
Affinity DataIC50: 112nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346506BDBM346506((2-cyanophenyl)methyl 4-(3-hydroxy-3-methyl-but-1-...)
Affinity DataIC50: 116nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346447BDBM346447(ethyl 4-[2-(3-aminophenyl)ethynyl]-2,6-dimethyl-7-...)
Affinity DataIC50: 120nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346509BDBM346509((2-methoxyphenyl)methyl-4-(3-hydroxy-3-methyl-but-...)
Affinity DataIC50: 123nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346522BDBM346522(isobutyl 4-(3-cyclopropyl-3-hydroxy-but-1-ynyl)-2,...)
Affinity DataIC50: 123nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346513BDBM346513(p-tolylmethyl 4-(3-hydroxy-3-methyl-but-1-ynyl)-2,...)
Affinity DataIC50: 128nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346556BDBM346556(isobutyl 4-(3-hydroxy-3-phenyl-but-1-ynyl)-2,6-dim...)
Affinity DataIC50: 130nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346425BDBM346425(ethyl 4-[(3R)-3-hydroxy-3-(5-methylisoxazol-3-yl)b...)
Affinity DataIC50: 136nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346575BDBM346575(4-(3-cyclopropyl-3-hydroxy-but-1-ynyl)-3-(5-isobut...)
Affinity DataIC50: 137nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346422BDBM346422(ethyl 4-(4-cyano-3-hydroxy-3-methyl-but-1-ynyl)-2,...)
Affinity DataIC50: 139nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346515BDBM346515((2-fluorophenyl)methyl 4-(3-hydroxy-3-methyl-but-1...)
Affinity DataIC50: 145nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346404BDBM346404(ethyl 4-[3-(3-cyanophenyl)-3-hydroxy-but-1-ynyl]-2...)
Affinity DataIC50: 146nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346550BDBM346550(isobutyl 4-(4-cyano-3-hydroxy-3-methyl-but-1-ynyl)...)
Affinity DataIC50: 150nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346499BDBM346499(Benzyl 4-(3-hydroxy-3-methyl-but-1-ynyl)-2,6-dimet...)
Affinity DataIC50: 151nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346464BDBM346464(US10202378, Example 77 | US10202378, Example 92a |...)
Affinity DataIC50: 154nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346538BDBM346538(1,2-dimethylpropyl 4-[3-hydroxy-3-(5-methylisoxazo...)
Affinity DataIC50: 160nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346502BDBM346502([3-(hydroxymethyl)phenyl]methyl4-(3-cyclopropyl-3-...)
Affinity DataIC50: 166nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346514BDBM346514(m-tolylmethyl 4-(3-hydroxy-3-methyl-but-1-ynyl)-2,...)
Affinity DataIC50: 167nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346428BDBM346428(ethyl 2,6-dimethyl-7-oxo-4-[4,4,4-trifluoro-3-hydr...)
Affinity DataIC50: 171nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346528BDBM346528(isobutyl 4-(3-hydroxy-3-methyl-but-1-ynyl)-2,6-dim...)
Affinity DataIC50: 173nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346476BDBM346476(US10202378, Example 89 | US10202378, Example 93b |...)
Affinity DataIC50: 176nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346441BDBM346441(isobutyl 4-[(3R)-3-hydroxy-3-(5-methylisoxazol-3-y...)
Affinity DataIC50: 179nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346488BDBM346488(US10202378, Example 96a | 4-(3-cyclopropyl-3-hydro...)
Affinity DataIC50: 182nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346408BDBM346408(ethyl 4-(3-hydroxy-3-methyl-5-phenyl-pent-1-ynyl)-...)
Affinity DataIC50: 182nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346460BDBM346460(US10202378, Example 73 | US10202378, Example 91b |...)
Affinity DataIC50: 184nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346592BDBM346592(ethyl 4-[3-(3-carbamoylphenyl)-4,4,4-trifluoro-3-h...)
Affinity DataIC50: 185nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346496BDBM346496(ethyl 2,6-dimethyl-7-oxo-4-[4,4,4-trifluoro-3-hydr...)
Affinity DataIC50: 189nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346484BDBM346484(US10202378, Example 94a | US10202378, Example 94b ...)
Affinity DataIC50: 192nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346450BDBM346450(ethyl 4-[2-(3-hydroxyphenyl)ethynyl]-2,6-dimethyl-...)
Affinity DataIC50: 195nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346577BDBM346577(4-(3-cyclopropyl-3-hydroxy-but-1-ynyl)-3-(5-ethyl-...)
Affinity DataIC50: 199nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346490BDBM346490(US10202378, Example 97a | US10202378, Example 185 ...)
Affinity DataIC50: 205nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346388BDBM346388(ethyl 4-[3-[4-(dimethylamino)phenyl]-4,4,4-trifluo...)
Affinity DataIC50: 209nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346456BDBM346456(ethyl 4-[(3R)-3-hydroxy-3-(3-methylisoxazol-5-yl)b...)
Affinity DataIC50: 210nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346486BDBM346486(US10202378, Example 95a | 3-[5-[(dimethylamino)met...)
Affinity DataIC50: 211nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346401BDBM346401(ethyl 4-(3-hydroxy-3-methyl-4-phenyl-but-1-ynyl)-2...)
Affinity DataIC50: 212nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346562BDBM346562(2-cyanoethyl 2,6-dimethyl-7-oxo-4-(4,4,4-trifluoro...)
Affinity DataIC50: 214nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346492BDBM346492(US10202378, Example 98a | US10202378, Example 98b ...)
Affinity DataIC50: 216nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346420BDBM346420(ethyl 4-[3-(3-fluorophenyl)-3-hydroxy-but-1-ynyl]-...)
Affinity DataIC50: 218nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346547BDBM346547(1,1-dimethylpropyl 4-(3-hydroxy-3-methyl-but-1-yny...)
Affinity DataIC50: 221nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346530BDBM346530((2-cyano-1,1-dimethyl-ethyl)-4-(3-cyclopropyl-3-hy...)
Affinity DataIC50: 222nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346505BDBM346505(thiazol-2-ylmethyl 4-(3-cyclopropyl-3-hydroxy-but-...)
Affinity DataIC50: 222nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 346431BDBM346431(ethyl 2,6-dimethyl-7-oxo-4-[4,4,4-trifluoro-3-hydr...)
Affinity DataIC50: 226nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

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