Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase receptor UFO [473-894,Q764R]'
LigandChemical structure of BindingDB Monomer ID 588269BDBM588269(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyazetidi...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588271BDBM588271(1-N'-(4-fluorophenyl)-1-N-[4-(7- methoxy-6-pyridin...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605730BDBM605730(US11673897, Compound 82 | l-N'-[6-[(6,7-dimethoxy-...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588252BDBM588252(1-N-[4-(7-carbamoylquinolin- 4-yl)oxyphenyl]-1-N'-...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588273BDBM588273(1-N'-(4-fluorophenyl)-1-N-[4-(7- methoxy-6-sulfamo...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588244BDBM588244(1-N-[4-(7-carbamoyl-6- methylquinolin-4-yl)oxyphen...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588223BDBM588223(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2S)...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588222BDBM588222(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2R)...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605727BDBM605727(US11673897, Compound 60 | 1-N-(4-fluorophenyl)-1-N...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588266BDBM588266(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyoxetan-...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605726BDBM605726(US11673897, Compound 18 | 1-N'-[6-(6-carbamoyl-7- ...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588225BDBM588225(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(1,3-ox...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588216BDBM588216(1-N'-(4-fluorophenyl)-N-[4-[7- methoxy-6-(2-piperi...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588237BDBM588237(1-N'-[3-chloro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605720BDBM605720(US11673897, Compound 10 | methyl 4-[5-[[1-[(4- flu...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588238BDBM588238(methyl 4-[2-fluoro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588217BDBM588217(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(2-morp...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588240BDBM588240(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605721BDBM605721(US11673897, Compound 11 | methyl 4-[3-chloro-5-[[1...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588263BDBM588263(1-N-[4-(6-cyclopropyl-7- methoxyquinolin-4- yl)oxy...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588241BDBM588241(1-N'-[3-fluoro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588232BDBM588232(1-N-[4-[6-carbamoyl-7-(3- morpholin-4- ylpropoxy)q...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588275BDBM588275(1-N'-(4-fluorophenyl)-1-N-[4-[7- methoxy-6-(1,3,4-...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588274BDBM588274(1-N'-(4-fluorophenyl)-1-N-[4-(7- methoxy-6- methyl...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588253BDBM588253(1-N'-(4-fluorophenyl)-1-N-[4- [7-(methylcarbamoyl)...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588255BDBM588255(1-N'-(4-fluorophenyl)-1-N-[4-(7- methoxy-6-pyridin...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588234BDBM588234(methyl 4-[2-chloro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588213BDBM588213(1-N-[4-(6-carbamoyl-7- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588236BDBM588236(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588214BDBM588214(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (methy...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588248BDBM588248(1-N-[4-(7-carbamoyl-6- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588227BDBM588227(1-N'-(4-fluorophenyl)-1-N- [4-[6- (methylcarbamoyl...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588226BDBM588226(1-N-[4-(6-carbamoylquinolin- 4-yl)oxyphenyl]-1-N'-...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605729BDBM605729(US11673897, Compound 81 | 1-N'-[6-[(6,7-dimethoxy-...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588228BDBM588228(1-N'-(4-fluorophenyl)-1-N- [4-[6-[(1-methylazetidi...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588270BDBM588270(1-N-[4-[6-(3,3-difluoroazetidin- 1-yl)-7-methoxyqu...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588249BDBM588249(1-N'-(4-fluorophenyl)-1-N- [4-[6-methoxy-7- (methy...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588272BDBM588272(1-N'-(4-fluorophenyl)-1-N-[4-(7- methoxy-6-pyridin...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588250BDBM588250(methyl 4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cycl...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588229BDBM588229(1-N-[4-(6-carbamoyl-7- fluoroquinolin-4-yl)oxyphen...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588264BDBM588264(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (1H-py...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605724BDBM605724(US11673897, Compound 16 | 1-N'-[6-(6-carbamoyl-7- ...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588242BDBM588242(methyl 4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cycl...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588221BDBM588221(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyazetidi...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 605725BDBM605725(US11673897, Compound 17 | 1-N-(4-fluorophenyl)-1-N...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEQ ID NO. 43), 10 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588265BDBM588265(tert-butyl 3-[4-[4-[[1-[(4- fluorophenyl)carbamoyl...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588224BDBM588224(1-N-[4-(6-cyano-7- methoxyquinolin-4- yl)oxyphenyl...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588267BDBM588267(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyazetidi...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588245BDBM588245(1-N'-(4-fluorophenyl)-1-N- [4-[6-methyl-7- (methyl...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588268BDBM588268(1-N-[4-[6-(azetidin-1-yl)-7- methoxyquinolin-4- yl...)
Affinity DataIC50: 55nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

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