Affinity DataKi: 0.0300nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris X33 using KHLY-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Inhibition of rat mast cell chymase using Suc-AAPF-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of KLK4 (unknown origin) expressed in Sf9 cells using FVQRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to RXRgammaMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to RXRbetaMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris X33 using KHLY-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of KLK4 (unknown origin) expressed in Sf9 cells using FVQRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to RXRbetaMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of recombinant human matriptase using Boc-QAR-MCA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity to RXRgammaMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity to RXRbetaMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity to RXRgammaMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to RXRgammaMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to RXRbetaMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity to RXRbetaMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Inhibition of recombinant KLK7 (unknown origin) expressed in zymogen form in Pichia pastorisstrain X-33 using KHLY-pNA as substrate after 30 minsMore data for this Ligand-Target Pair