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Found 332 with Last Name = 'green' and Initial = 'dw'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037121(2-[(1R,3S,4S)-1-BENZYL-4-[N-(BENZYLOXYCARBONYL)-L-...)
Affinity DataKi:  0.600nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037124((R)-2-{(R)-2-[(S)-4-((S)-2-Benzyloxycarbonylamino-...)
Affinity DataKi:  0.700nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037122(CHEMBL108016 | [(1S,2S,4R)-1-Benzyl-2-hydroxy-4-(5...)
Affinity DataKi:  83nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037126(CHEMBL80098 | [(1S,2S,4R)-1-Benzyl-2-hydroxy-5-phe...)
Affinity DataKi:  92nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037125(CHEMBL107849 | {(S)-1-Benzyl-4-[(S)-1-(carbamoylme...)
Affinity DataKi:  120nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037128(CHEMBL419921 | [(1S,2S,4R)-1-Benzyl-4-(5-butyryl-1...)
Affinity DataKi:  150nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037123(CHEMBL108226 | {(1S,2S,4R)-1-Benzyl-4-[5-(2,2-dime...)
Affinity DataKi:  270nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037127(CHEMBL104285 | [(1S,2S,4R)-4-(5-Acetyl-1H-imidazol...)
Affinity DataKi:  370nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032937(2-{2-[(S)-2-(3-Benzyl-5-{1-[(1-carboxy-ethyl)-meth...)
Affinity DataKi:  430nMAssay Description:Competitive inhibitory activity of the compound was determined against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037120(CHEMBL104523 | {(1S,2S,4R)-1-Benzyl-2-hydroxy-4-[5...)
Affinity DataKi:  2.70E+3nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037129(CHEMBL106776 | [(1S,2S,4R)-1-Benzyl-4-(5-formyl-1H...)
Affinity DataKi:  3.50E+3nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50037119(CHEMBL448480 | {(1S,2S,4R)-1-Benzyl-2-hydroxy-4-[5...)
Affinity DataKi:  1.33E+4nMAssay Description:Apparent inhibition constant against recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032938(2-{2-[(S)-2-(3-Benzyl-5-{1-[(1-carboxy-ethyl)-meth...)
Affinity DataKi:  1.47E+5nMAssay Description:Competitive inhibitory activity of the compound was determined against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375120(CHEMBL403040)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142256(4-(4-tert-Butyl-benzenesulfonyl)-1-(3H-imidazol-4-...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0-ATP synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375119(CHEMBL401868)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375121(CHEMBL257038)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375116(CHEMBL403290)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375124(CHEMBL256457)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375116(CHEMBL403290)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375116(CHEMBL403290)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375121(CHEMBL257038)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375119(CHEMBL401868)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375123(CHEMBL272558)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375122(CHEMBL427833)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375117(CHEMBL255798)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375122(CHEMBL427833)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375116(CHEMBL403290)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375120(CHEMBL403040)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375111(CHEMBL409499)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142274(4-(3,4-Dichloro-benzenesulfonyl)-1-(5-methyl-3H-im...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0-ATP hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50371837(CHEMBL257663)
Affinity DataIC50:  30nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50371837(CHEMBL257663)
Affinity DataIC50:  30nMAssay Description:Displacement of [125]CXCL10 from human CXCR3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50404297(CHEMBL269080)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0 ATP hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375117(CHEMBL255798)
Affinity DataIC50:  30nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50404288(CHEMBL269369)
Affinity DataIC50:  33nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0-ATP synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50404288(CHEMBL269369)
Affinity DataIC50:  33nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0 ATP hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142256(4-(4-tert-Butyl-benzenesulfonyl)-1-(3H-imidazol-4-...)
Affinity DataIC50:  38nMAssay Description:Inhibitory activity of the compound against ccytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375120(CHEMBL403040)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]-CXCL10 from mouse CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375124(CHEMBL256457)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375123(CHEMBL272558)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375122(CHEMBL427833)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]-CXCL10 from mouse CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375121(CHEMBL257038)
Affinity DataIC50:  60nMAssay Description:Displacement of [125I]-CXCL10 from mouse CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375126(CHEMBL255583)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cell membrane assessed as inhibition of calcium flux by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375116(CHEMBL403290)
Affinity DataIC50:  70nMAssay Description:Displacement of [125I]-CXCL10 from mouse CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50371837(CHEMBL257663)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by FLIPR-based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142258(4-(4-tert-Butyl-benzenesulfonyl)-1-(5-methyl-3H-im...)
Affinity DataIC50:  77nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0-ATP hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50404319(CHEMBL266556)
Affinity DataIC50:  77nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0-ATP synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit beta,/delta,/epsilon,/gamma, mitochondrial(Bos taurus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50404307(CHEMBL8366)
Affinity DataIC50:  77nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0-ATP hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Abbott Bioresearch Center

Curated by ChEMBL
LigandPNGBDBM50375116(CHEMBL403290)
Affinity DataIC50:  80nMAssay Description:Displacement of [125I]-CXCL10 from mouse CXCR3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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