Affinity DataKi: 49nMAssay Description:Competitive antagonist activity at human P2X4 receptor expressed in 1321N1 cell membrane assessed as inhibition of [35S]ATPgammaS binding by scintill...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetLeucine--tRNA ligase, cytoplasmic(Saccharomyces cerevisiae S288c)
Anacor Pharmaceuticals
Curated by ChEMBL
Anacor Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.85E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae cytoplasmic leucyl-tRNA synthetase after 20 minsMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Frankfurt
Curated by ChEMBL
Goethe-University Frankfurt
Curated by ChEMBL
Affinity DataKi: 4.80E+3nMAssay Description:Competitive inhibition of full length human soluble epoxide hydrolase pre-incubated for 30 mins before DiFMUP substrate addition by fluorescence base...More data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Goethe-University Frankfurt
Curated by ChEMBL
Goethe-University Frankfurt
Curated by ChEMBL
Affinity DataKi: 4.80E+3nMAssay Description:Competitive inhibition of full length human soluble epoxide hydrolase pre-incubated for 30 mins before DiFMUP substrate addition by fluorescence base...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetLeucine--tRNA ligase, cytoplasmic(Saccharomyces cerevisiae S288c)
Anacor Pharmaceuticals
Curated by ChEMBL
Anacor Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.14E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae cytoplasmic leucyl-tRNA synthetase after 2 minsMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.40E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.90E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4.90E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 7.80E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 8.10E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 9.10E+4nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.90E+5nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human placental cytosolic 17beta-HSD1 using [3H]-E1 as substrate after 10 mins in presence of NADPH by radio-flow detector based analys...More data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human placental cytosolic 17beta-HSD1 using [3H]-E1 as substrate after 10 mins in presence of NADPH by radio-flow detector based analys...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human placental cytosolic 17beta-HSD1 using [3H]-E1 as substrate after 10 mins in presence of NADPH by radio-flow detector based analys...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human placental cytosolic 17beta-HSD1 using [3H]-E1 as substrate after 10 mins in presence of NADPH by radio-flow detector based analys...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human placental microsomal fraction 17beta-HSD2 using [3H]-E2 as substrate after 20 mins in presence of NAD+ by radio-flow detector bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human placental cytosolic 17beta-HSD1 using [3H]-E1 as substrate after 10 mins in presence of NADPH by radio-flow detector based analys...More data for this Ligand-Target Pair