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Found 66 with Last Name = 'shantharam' and Initial = 'cs'
TargetAlpha-galactosidase(Coffea arabica (Coffee beans))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50520994(CHEMBL4529797)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of green coffee bean alpha-galactosidaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50520989(CHEMBL4565280)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of human recombinant FTase using [3H]FPP as substrate after 15 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM11823(Azepane Derivative 4 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of PKBalpha (unknown origin) expressed in Sf9 insect cells using Biotin-SGRARTSSFAEPG as substrate after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  12.7nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50526706(CHEMBL4545676)
Affinity DataIC50:  270nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM222462((E)-4-[4-(2-Chlorobenzylidene)-2-(4-chlorophenyl)-...)
Affinity DataIC50:  860nMAssay Description:Inhibition of recombinant human COX2 by EIAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50520992(CHEMBL4438366)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of beta-galactosidase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425942(CHEMBL2313740)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425923(CHEMBL2313709)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425946(CHEMBL2313736)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425911(CHEMBL2313700)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50502118(CHEMBL4476702)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-a-d-glucopyranoside as substrate preincubated for 5 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425932(CHEMBL2313729)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425927(CHEMBL2313705)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425934(CHEMBL2313727)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425910(CHEMBL2313701)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425912(CHEMBL2313699)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425921(CHEMBL2313711)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425913(CHEMBL2313698)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM222462((E)-4-[4-(2-Chlorobenzylidene)-2-(4-chlorophenyl)-...)
Affinity DataIC50:  7.86E+3nMAssay Description:Inhibition of ovine COX1 by EIAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425931(CHEMBL2313730)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425940(CHEMBL2313719)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425933(CHEMBL2313728)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50512315(CHEMBL4438040)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) aggregationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM192670(3-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-1-(4-o-...)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425944(CHEMBL2313738)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM192678(1-(4-(3-chlorophenyl)piperazin-1-yl)-3-(6-methoxy-...)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425943(CHEMBL2313739)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425947(CHEMBL2313735)
Affinity DataIC50:  2.02E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425925(CHEMBL2313707)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Aspergillus oryzae)
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50520993(CHEMBL4472415)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Aspergillus oryzae beta-galactosidaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425945(CHEMBL2313737)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425924(CHEMBL2313708)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM192669(3-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-1-(4-ph...)
Affinity DataIC50:  2.42E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Homo sapiens (Human))
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM178133(3-(6-Chloro-1H-imidazo[4,5-b]pyridin-2-yl)benzene-...)
Affinity DataIC50:  2.93E+4nMAssay Description:Inhibition of beta-glucuronidase (unknown origin) using p-nitrophenyl-beta-D-glucuronide as substrate pre-incubated for 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425928(CHEMBL2313704)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425926(CHEMBL2313706)
Affinity DataIC50:  3.34E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50217942(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chr...)
Affinity DataIC50:  4.19E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425922(CHEMBL2313710)
Affinity DataIC50:  5.48E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425941(CHEMBL2313718)
Affinity DataIC50:  5.55E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425914(CHEMBL2313697)
Affinity DataIC50:  5.94E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425915(CHEMBL2313717)
Affinity DataIC50:  6.03E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425937(CHEMBL2313722)
Affinity DataIC50:  7.03E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425918(CHEMBL2313714)
Affinity DataIC50:  7.09E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425938(CHEMBL2313721)
Affinity DataIC50:  7.58E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425919(CHEMBL2313713)
Affinity DataIC50:  7.61E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425935(CHEMBL2313725)
Affinity DataIC50:  8.39E+4nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425939(CHEMBL2313720)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425920(CHEMBL2313712)
Affinity DataIC50:  1.17E+5nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Bos taurus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50425916(CHEMBL2313716)
Affinity DataIC50:  1.26E+5nMAssay Description:Inhibition of glycation of bovine serum albumin assessed as advanced glycated end product measured after 7 days by spectrofluorimeter in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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