Report error Found 1000 Enz. Inhib. hit(s) with Target = 'Synaptic vesicular amine transporter'
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Binding affinity to VMAT2More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal membrane homogenatesMore data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Displacement of [3H]-DTBZ from VMAT2 in rat striatal membrane homogenatesMore data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.520nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.680nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.820nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.930nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of dopamine uptake at VMAT in bovine chromaffin granule ghostsMore data for this Ligand-Target Pair
Affinity DataKi: 1.03nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Examples of techniques for determining the capability of a compound to inhibit VMAT2 are provided below. The procedure is adapted from that described...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Examples of techniques for determining the capability of a compound to inhibit VMAT2 are provided below. The procedure is adapted from that described...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Examples of techniques for determining the capability of a compound to inhibit VMAT2 are provided below. The procedure is adapted from that described...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
Affinity DataKi: 2.45nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal membrane homogenatesMore data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Examples of techniques for determining the capability of a compound to inhibit VMAT2 are provided below. The procedure is adapted from that described...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Examples of techniques for determining the capability of a compound to inhibit VMAT2 are provided below. The procedure is adapted from that described...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Examples of techniques for determining the capability of a compound to inhibit VMAT2 are provided below. The procedure is adapted from that described...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Examples of techniques for determining the capability of a compound to inhibit VMAT2 are provided below. The procedure is adapted from that described...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Human)
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:The human VMAT2 Ki values for the compounds listed in Table 15A and Table 15B were determined using the following procedures. Compound dilution serie...More data for this Ligand-Target Pair
Affinity DataKi: 3.75nMAssay Description:Displacement of [3H]-DTBZ from VMAT2 in rat striatal membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 3.96nMAssay Description:Displacement of [3H]DHTBZ from Sprague-Dawley rat striatum VMAT2 after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of dopamine uptake at VMAT in bovine chromaffin granule ghostsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition constant against [3H]-nicotine binding to vesicular monoamine transporter-2 of rat brain membranesMore data for this Ligand-Target Pair
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