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Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 2892
TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25891((2S)-2-[(5-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50:  25nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25890((2S)-2-[(5-formylthiophen-2-yl)formamido]-3-methyl...)
Affinity DataIC50:  85nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25892((2S)-2-[(4-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50:  100nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25889((2S)-2-[(5-formylfuran-2-yl)formamido]-3-methyl-N-...)
Affinity DataIC50:  100nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25887((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50:  100nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25894((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50:  110nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25886((2S)-2-(furan-2-ylformamido)-3-methyl-N-[(2S)-4-me...)
Affinity DataIC50:  135nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25895(N-heterocyclic dipeptide aldehyde, 13 | methyl 5-{...)
Affinity DataIC50:  140nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25893((2S)-2-[(5-formyl-1-methyl-1H-pyrrol-2-yl)formamid...)
Affinity DataIC50:  150nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25893((2S)-2-[(5-formyl-1-methyl-1H-pyrrol-2-yl)formamid...)
Affinity DataIC50:  150nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25891((2S)-2-[(5-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50:  290nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25895(N-heterocyclic dipeptide aldehyde, 13 | methyl 5-{...)
Affinity DataIC50:  290nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetCalpain-2 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25888((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50:  315nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25894((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50:  340nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25890((2S)-2-[(5-formylthiophen-2-yl)formamido]-3-methyl...)
Affinity DataIC50:  440nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25892((2S)-2-[(4-formyl-1H-pyrrol-2-yl)formamido]-3-meth...)
Affinity DataIC50:  530nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25888((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50:  650nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25887((2S)-3-methyl-N-[(2S)-4-methyl-1-oxopentan-2-yl]-2...)
Affinity DataIC50:  680nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25886((2S)-2-(furan-2-ylformamido)-3-methyl-N-[(2S)-4-me...)
Affinity DataIC50:  790nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCalpain-1 catalytic subunit(Sheep)
University of Canterbury

LigandPNGBDBM25889((2S)-2-[(5-formylfuran-2-yl)formamido]-3-methyl-N-...)
Affinity DataIC50:  960nMpH: 7.5 T: 25°CAssay Description:Calpain inhibition assays were performed in 96-well black plates. The reaction was initiated by the addition of substrate solution. The progress of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed