Compile Data Set for Download or QSAR
Report error Found 101 Enz. Inhib. hit(s) with all data for entry = 50027780
TargetCollagenase 3(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-16(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 0.310nMAssay Description:Inhibition of MMP16More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273426(N-(4-Phenoxybenzenesulfonyl)-N-hydroxycarbonylmeth...)
Affinity DataIC50: 0.330nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273426(N-(4-Phenoxybenzenesulfonyl)-N-hydroxycarbonylmeth...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273426(N-(4-Phenoxybenzenesulfonyl)-N-hydroxycarbonylmeth...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241252(2-[hydroxycarbamoylmethyl-(4-phenoxy-benzenesulfon...)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241252(2-[hydroxycarbamoylmethyl-(4-phenoxy-benzenesulfon...)
Affinity DataIC50: 0.740nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273426(N-(4-Phenoxybenzenesulfonyl)-N-hydroxycarbonylmeth...)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-16(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241252(2-[hydroxycarbamoylmethyl-(4-phenoxy-benzenesulfon...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP16More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246601(2-(N-(2-(hydroxyamino)-2-oxoethyl)-4-phenoxyphenyl...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-16(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273426(N-(4-Phenoxybenzenesulfonyl)-N-hydroxycarbonylmeth...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of MMP16More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246601(2-(N-(2-(hydroxyamino)-2-oxoethyl)-4-phenoxyphenyl...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241252(2-[hydroxycarbamoylmethyl-(4-phenoxy-benzenesulfon...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241252(2-[hydroxycarbamoylmethyl-(4-phenoxy-benzenesulfon...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246601(2-(N-(2-(hydroxyamino)-2-oxoethyl)-4-phenoxyphenyl...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246601(2-(N-(2-(hydroxyamino)-2-oxoethyl)-4-phenoxyphenyl...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241250(N-(4-Biphenylsulfonyl)-N-{[2-(4-sulfamoylphenyl)et...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273426(N-(4-Phenoxybenzenesulfonyl)-N-hydroxycarbonylmeth...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of human recombinant CA2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273425(N-(4-Biphenylsulfonyl)-N-hydroxycarbonylmethyl-D-v...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50066658((R)-N-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-pyrid...)
Affinity DataIC50: 5nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM11635(4-sulfamoyl-N-[2-(4-sulfamoylphenyl)ethyl]benzamid...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant CA2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50066658((R)-N-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-pyrid...)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241249(((4-phenoxy-benzenesulfonyl)-{[2-(4sulfamoyl-pheny...)
Affinity DataKi:  6.40nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-16(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50066658((R)-N-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-pyrid...)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of MMP16More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50066658((R)-N-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-pyrid...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246599(N-(4-Phenoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241250(N-(4-Biphenylsulfonyl)-N-{[2-(4-sulfamoylphenyl)et...)
Affinity DataKi:  8.40nMAssay Description:Inhibition of human recombinant CA2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241249(((4-phenoxy-benzenesulfonyl)-{[2-(4sulfamoyl-pheny...)
Affinity DataKi:  9.30nMAssay Description:Inhibition of human recombinant CA2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-16(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246601(2-(N-(2-(hydroxyamino)-2-oxoethyl)-4-phenoxyphenyl...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MMP16More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241252(2-[hydroxycarbamoylmethyl-(4-phenoxy-benzenesulfon...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant CA2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241253(2-[(biphenyl-4-sulfonyl)-hydroxycarbamoylmethyl-am...)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241251(N-(4-Methoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50246601(2-(N-(2-(hydroxyamino)-2-oxoethyl)-4-phenoxyphenyl...)
Affinity DataIC50: 14nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241253(2-[(biphenyl-4-sulfonyl)-hydroxycarbamoylmethyl-am...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM11635(4-sulfamoyl-N-[2-(4-sulfamoylphenyl)ethyl]benzamid...)
Affinity DataKi:  18nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50066658((R)-N-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-pyrid...)
Affinity DataIC50: 23nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50066658((R)-N-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-pyrid...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  25nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241251(N-(4-Methoxybenzenesulfonyl)-N-{[2-(4-sulfamoylphe...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273425(N-(4-Biphenylsulfonyl)-N-hydroxycarbonylmethyl-D-v...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant MMP2 transfected in mouse melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50241254(2-(benzyl-hydroxycarbamoylmethyl-amino)-N-[2-(4-su...)
Affinity DataKi:  26nMAssay Description:Inhibition of human recombinant CA9 catalytic domain by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273425(N-(4-Biphenylsulfonyl)-N-hydroxycarbonylmethyl-D-v...)
Affinity DataIC50: 28nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Instituto Superior TéCnico

Curated by ChEMBL
LigandPNGBDBM50273424(N-(4-Methoxybenzenesulfonyl)-N-hydroxycarbonylmeth...)
Affinity DataIC50: 29nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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