Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 9568
TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475864(2-(4-((3-(2′-(difluoromethoxy)-2,6-dimethyl-...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475863(2-(4-((3-(2,6-dichloro-2′-(difluoromethoxy)-...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441830(US10647665, Example 1-17 | US10851050, Example I-1...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441829(US10647665, Example 1-16 | US10851050, Example I-1...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441828(US10647665, Example 1-15 | US10851050, Example I-1...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441825(US10647665, Example 1-13 | US10851050, Example I-1...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441823(US10647665, Example 1-12 | US10851050, Example I-1...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441822(US10647665, Example 1-11 | US10851050, Example I-1...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441820(US10647665, Example 1-9 | US10851050, Example I-9)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475882(2-(4-((3-(2,6-dichloro-2′-(trifluoromethoxy)...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441818(US10647665, Example 1-7 | US10851050, Example I-7)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475881(2-(4-((3-(2,6-dichloro-2′-(trifluoromethoxy)...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441817(US10647665, Example 1-6 | US10851050, Example I-6)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441816(US10647665, Example 1-5 | US10851050, Example I-5)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475879(3-(4-((3-(2,6-dichloro-2′-(trifluoromethoxy)...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441815(US10647665, Example 1-4 | US10851050, Example I-4)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475878(3-(4-((3-(2,6-dichloro-2′-(trifluoromethoxy)...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475877(3-(4-((3-(2,6-dichloro-2′-(trifluoromethoxy)...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475876(3-(4-((3-(2,6-dichloro-2′-(trifluoromethoxy)...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441846(US10647665, Example 1-35 | US10647665, Example 1-3...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441843(US10647665, Example 1-29 | US10851050, Example I-2...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441839(US10647665, Example 1-25 | US10851050, Example I-2...)
Affinity DataIC50: 500nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441838(US10647665, Example 1-24 | US10851050, Example I-2...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441836(US10647665, Example 1-22b | US10851050, Example I-...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441835(US10647665, Example 1-22a | US10851050, Example I-...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441832(US10647665, Example 1-19 | US10851050, Example I-1...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441831(US10647665, Example 1-18 | US10851050, Example I-1...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441827(US10647665, Example 1-14 | US10851050, Example I-1...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441821(US10647665, Example 1-10 | US10851050, Example I-1...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441819(US10647665, Example 1-8 | US10851050, Example I-8)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM475880(3-(4-((3-(2,6-dichloro-2′-(trifluoromethoxy)...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441814(US10647665, Example 1-3 | US10851050, Example I-3)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441845(US10647665, Example 1-31 | US10851050, Example I-3...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441844(US10647665, Example 1-30 | US10851050, Example I-3...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441842(US10647665, Example 1-28 | US10851050, Example I-2...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441841(US10647665, Example 1-27 | US10851050, Example I-2...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441840(US10647665, Example 1-26 | US10851050, Example I-2...)
Affinity DataIC50: 2.75E+3nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441837(US10647665, Example 1-23 | US10851050, Example I-2...)
Affinity DataIC50: 2.75E+4nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Fudan University

US Patent
LigandPNGBDBM441813(US10647665, Example 1-2 | US1085105, Example I-2)
Affinity DataIC50: 2.75E+4nMAssay Description:The inhibitory activity of compounds on RORγ receptor was determined by fluorescence resonance energy transfer (FRET) experiments. The inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2021
Entry Details
US Patent