Compile Data Set for Download or QSAR
Report error Found 135 Enz. Inhib. hit(s) with all data for entry = 9824
TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373616BDBM373616(US10246442, Example 69 | 1-(6-(4-Chlorophenoxy)-4-...)
Affinity DataIC50: 20nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373637BDBM373637(US10246442, Example 83 | 1-(4-(Diethylamino)-7-phe...)
Affinity DataIC50: 20nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373609BDBM373609(US10246442, Example 63 | 1-(6-(4-Chlorophenoxy)-4-...)
Affinity DataIC50: 25.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373661BDBM373661(US10246442, Example 102 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 31.6nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373612BDBM373612(US10246442, Example 66 | 1-(4-(Azepan-1-yl)-6-(4-c...)
Affinity DataIC50: 31.6nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373610BDBM373610(US10246442, Example 64 | 1-(6-(4-Chlorophenoxy)-4-...)
Affinity DataIC50: 31.6nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373668BDBM373668(US10246442, Example 138 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 31.6nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373563BDBM373563(US10246442, Example 24 | 1-(4-Amino-6-cyclohexylqu...)
Affinity DataIC50: 31.6nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373544BDBM373544(US10246442, Example 6 | 1-[6-(2,6-Dimethyl-phenoxy...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373543BDBM373543(US10246442, Example 5 | 1-[6-(2,6-Dimethyl-phenoxy...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373676BDBM373676(US10246442, Example 164 | 1-(4-(Ethyl(methyl)amino...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373673BDBM373673(US10246442, Example 161 | 1-(4-(Dimethylamino)-7-c...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373611BDBM373611(US10246442, Example 65 | 1-(6-(4-chlorophenoxy)-4-...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373589BDBM373589(US10246442, Example 46 | 1-(4-(Diethylamino)-6-phe...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373627BDBM373627(US10246442, Example 77 | 1-(4-(Dimethylamino)-7-ph...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373550BDBM373550(US10246442, Example 12 | 1-[6-(2,6-Dimethyl-phenox...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373667BDBM373667(US10246442, Example 137 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373679BDBM373679(US10246442, Example 173 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 39.8nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373675BDBM373675(US10246442, Example 163 | 1-(7-Chloro-6-isopropyl-...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373613BDBM373613(US10246442, Example 67 | 1-(6-(4-Chlorophenoxy)-4-...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373631BDBM373631(US10246442, Example 78 | 1-(7-Phenoxy-4-(pyrrolidi...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 50446891BDBM50446891(CHEMBL3115314 | US10246442, Example 61 | US1097506...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373569BDBM373569(US10246442, Example 28 | 1-(6-Cyclohexyl-4-(phenyl...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373605BDBM373605(US10246442, Example 60 | 1-(6-(4-Chlorophenoxy)-4-...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373684BDBM373684(US10246442, Example 177 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373568BDBM373568(US10246442, Example 27 | 1-(6-Cyclohexyl-4-(diethy...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373586BDBM373586(US10246442, Example 43 | 1-(6-Phenyl-4-(pyrrolidin...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373622BDBM373622(US10246442, Example 74 | 1-(4-(Diethylamino)-6-phe...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373585BDBM373585(US10246442, Example 42 | 1-(4-(Ethyl(methyl)amino)...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373662BDBM373662(US10246442, Example 103 | 1-(6-(Cyclohexyloxy)-7-f...)
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373674BDBM373674(US10246442, Example 162 | 1-(4-(Diethylamino)-7-ch...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373591BDBM373591(US10246442, Example 48 | 1-(4-(Azepan-1-yl)-6-phen...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373553BDBM373553(US10246442, Example 15 | 1-((4-Cyclopropanemethyla...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373670BDBM373670(US10246442, Example 140 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373588BDBM373588(US10246442, Example 45 | 1-(6-Phenyl-4-(piperidin-...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373621BDBM373621(US10246442, Example 73 | 1-(6-Phenoxy-4-(pyrrolidi...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373665BDBM373665(US10246442, Example 105 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373584BDBM373584(US10246442, Example 41 | 1-(4-(Dimethylamino)-6-ph...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373546BDBM373546(US10246442, Example 8 | 1-[6-(2,6-Dimethyl-phenoxy...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373545BDBM373545(US10246442, Example 7 | 1-[4-(2-Chloro-phenylamino...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373581BDBM373581(US10246442, Example 38 | 1-(6-Cyclohexyl-4-(dimeth...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373541BDBM373541(US10246442, Example 3 | 1-[4-Dimethylamino-6-(2,6-...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373578BDBM373578(US10246442, Example 35 | 1-(4-Cyanamido-6-cyclohex...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373540BDBM373540(US10246442, Example 2 | 1-[6-(2,6-Dimethyl-phenoxy...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373691BDBM373691(US10246442, Example 183 | 1-(6-Benzyl-4-(ethyl(met...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373539BDBM373539(US10246442, Example 1 | 1-[4-Amino-6-(2,6-dimethyl...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373649BDBM373649(US10246442, Example 94 | 1-(4-(Ethyl(methyl)amino)...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373648BDBM373648(US10246442, Example 93 | 1-(4-(Dipropylamino)-7-ph...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373681BDBM373681(US10246442, Example 175 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetEgl nine homolog 1 [181-417](Human)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 373680BDBM373680(US10246442, Example 174 | 1-(6-(Cyclohexyloxy)-4-(...)
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

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