Compile Data Set for Download or QSAR
Report error Found 330 Enz. Inhib. hit(s) with all data for entry = 11095
TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142088BDBM142088(US8933056, Ala-boroPro Thioxamide | US11096924, DA...)
Affinity DataIC50: 0.200nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142088BDBM142088(US8933056, Ala-boroPro Thioxamide | US11096924, DA...)
Affinity DataIC50: 0.200nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050516BDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50: 0.200nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514526BDBM514526(US11096924, DASH-inhibitors 5362 | US11583516, Cmp...)
Affinity DataIC50: 0.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050525BDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 0.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050525BDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 0.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050513BDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 0.700nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050515BDBM50050515(Boronic acid derivative | CHEMBL63652 | US11096924...)
Affinity DataIC50: 0.800nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142092BDBM142092(US8933056, Val-boroPro Thioxamide | US11096924, DA...)
Affinity DataIC50: 0.800nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050527BDBM50050527(Boronic acid derivative | CHEMBL66032 | US11096924...)
Affinity DataIC50: 0.900nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514523BDBM514523(US11096924, DASH-inhibitors 2408 | US11559537, Com...)
Affinity DataIC50: 0.900nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050528BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
Affinity DataIC50: 1nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050525BDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 1nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142093BDBM142093(US8933056, Chg-boroPro Thioxamide | US8933056, Chg...)
Affinity DataIC50: 1.10nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50253621BDBM50253621((S)-4-amino-5-((R)-2-boronopyrrolidin-1-yl)-5-oxop...)
Affinity DataIC50: 1.10nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142093BDBM142093(US8933056, Chg-boroPro Thioxamide | US8933056, Chg...)
Affinity DataIC50: 1.20nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50369128BDBM50369128(CHEMBL1790483 | US11096924, DASH-inhibitors 4316 |...)
Affinity DataIC50: 1.20nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050521BDBM50050521((2R)-N-[(2R)-2-(DIHYDROXYBORYL)-1-L-PROLYLPYRROLID...)
Affinity DataIC50: 1.30nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050516BDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50: 1.30nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50151003BDBM50151003(CHEMBL1627303 | CHEMBL363250 | (S)-1-((S)-2-Amino-...)
Affinity DataIC50: 1.30nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514555BDBM514555(US11096924, DASH-inhibitors 4367 | US11583516, Cmp...)
Affinity DataIC50: 1.40nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050525BDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 1.40nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514554BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
Affinity DataIC50: 1.40nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514555BDBM514555(US11096924, DASH-inhibitors 4367 | US11583516, Cmp...)
Affinity DataIC50: 1.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050528BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
Affinity DataIC50: 1.60nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050520BDBM50050520(Boronic acid derivative | CHEMBL63406 | US11096924...)
Affinity DataIC50: 1.60nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050516BDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50: 1.60nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050513BDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 1.70nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050520BDBM50050520(Boronic acid derivative | CHEMBL63406 | US11096924...)
Affinity DataIC50: 1.90nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 8(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514540BDBM514540(US11096924, DASH-inhibitors 5320 | US11583516, Cmp...)
Affinity DataIC50: 1.90nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514550BDBM514550(US11096924, DASH-inhibitors 4312 | US11559537, Com...)
Affinity DataIC50: 2nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50369128BDBM50369128(CHEMBL1790483 | US11096924, DASH-inhibitors 4316 |...)
Affinity DataIC50: 2nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514518BDBM514518(US11096924, DASH-inhibitors 4317 | US11559537, Com...)
Affinity DataIC50: 2nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050515BDBM50050515(Boronic acid derivative | CHEMBL63652 | US11096924...)
Affinity DataIC50: 2nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142093BDBM142093(US8933056, Chg-boroPro Thioxamide | US8933056, Chg...)
Affinity DataIC50: 2.10nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514526BDBM514526(US11096924, DASH-inhibitors 5362 | US11583516, Cmp...)
Affinity DataIC50: 2.40nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 8(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142093BDBM142093(US8933056, Chg-boroPro Thioxamide | US8933056, Chg...)
Affinity DataIC50: 2.70nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 8/9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514515BDBM514515(US11096924, DASH-inhibitors 3102 C | US11583516, C...)
Affinity DataIC50: 2.70nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514516BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
Affinity DataIC50: 2.70nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142088BDBM142088(US8933056, Ala-boroPro Thioxamide | US11096924, DA...)
Affinity DataIC50: 2.80nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514516BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
Affinity DataIC50: 2.80nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 2(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050527BDBM50050527(Boronic acid derivative | CHEMBL66032 | US11096924...)
Affinity DataIC50: 2.90nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514520BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
Affinity DataIC50: 2.90nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 8(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 589767BDBM589767(US11559537, Compound 5322)
Affinity DataIC50: 3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050525BDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 514518BDBM514518(US11096924, DASH-inhibitors 4317 | US11559537, Com...)
Affinity DataIC50: 3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 142092BDBM142092(US8933056, Val-boroPro Thioxamide | US11096924, DA...)
Affinity DataIC50: 3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050525BDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 3.10nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050515BDBM50050515(Boronic acid derivative | CHEMBL63652 | US11096924...)
Affinity DataIC50: 3.10nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 50050521BDBM50050521((2R)-N-[(2R)-2-(DIHYDROXYBORYL)-1-L-PROLYLPYRROLID...)
Affinity DataIC50: 3.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

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