Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 11210
TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474233BDBM474233(5-[5-amino-7-(4-fluorophenyl)-2-[(3-fluoropyrid in...)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474223BDBM474223(2-(2,6-difluorobenzyl)-8-(2-(dimethylamino) pyridi...)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474222BDBM474222(5-(5-amino-2-(2,6-difluorobenzyl)-7-(4- fluorophen...)
Affinity DataIC50: 0.200nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474230BDBM474230(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474237BDBM474237(5-(5-amino-7-(3-chlorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474230BDBM474230(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474223BDBM474223(2-(2,6-difluorobenzyl)-8-(2-(dimethylamino) pyridi...)
Affinity DataIC50: 0.900nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474221BDBM474221(8-(2,6-dimethylpyridin-4-yl)-7-(4-fluoropheny1)- 2...)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474238BDBM474238(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (3-...)
Affinity DataIC50: 1.40nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474227BDBM474227(5-[5-amino-2-[(2,6-difluorophenyl)methyl]-7-(2 H-1...)
Affinity DataIC50: 1.40nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474234BDBM474234(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (4-...)
Affinity DataIC50: 1.70nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474222BDBM474222(5-(5-amino-2-(2,6-difluorobenzyl)-7-(4- fluorophen...)
Affinity DataIC50: 2.10nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474232BDBM474232(5-(5-amino-7-(4-(difluoromethyl)phenyl)-2-((3-f lu...)
Affinity DataIC50: 2.20nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474221BDBM474221(8-(2,6-dimethylpyridin-4-yl)-7-(4-fluoropheny1)- 2...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474221BDBM474221(8-(2,6-dimethylpyridin-4-yl)-7-(4-fluoropheny1)- 2...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474223BDBM474223(2-(2,6-difluorobenzyl)-8-(2-(dimethylamino) pyridi...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474233BDBM474233(5-[5-amino-7-(4-fluorophenyl)-2-[(3-fluoropyrid in...)
Affinity DataIC50: 2.80nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474224BDBM474224(5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] me...)
Affinity DataIC50: 2.80nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474230BDBM474230(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 2.80nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474228BDBM474228(2-((3-fluoropyridin-2-yl)methyl)-8-(imidazo[l,2- a...)
Affinity DataIC50: 3nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474232BDBM474232(5-(5-amino-7-(4-(difluoromethyl)phenyl)-2-((3-f lu...)
Affinity DataIC50: 3.40nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474229BDBM474229(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50: 3.40nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474241BDBM474241(2-[(3-fluoropyridin-2-yl)methyl]-8-[imidazo[l,2- a...)
Affinity DataIC50: 3.5nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474238BDBM474238(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (3-...)
Affinity DataIC50: 3.60nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474231BDBM474231(6-[[5-amino-7-(4-fluorophenyl)-8-[imidazo[1,2-a] p...)
Affinity DataIC50: 4nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474224BDBM474224(5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] me...)
Affinity DataIC50: 4nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474233BDBM474233(5-[5-amino-7-(4-fluorophenyl)-2-[(3-fluoropyrid in...)
Affinity DataIC50: 4nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474237BDBM474237(5-(5-amino-7-(3-chlorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 4.10nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474234BDBM474234(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (4-...)
Affinity DataIC50: 4.20nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474235BDBM474235(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (4-...)
Affinity DataIC50: 5.10nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474235BDBM474235(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (4-...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474239BDBM474239(2-(2,6-difluorobenzyl)-8-(2-(difluoromethoxy) pyri...)
Affinity DataIC50: 5.40nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474239BDBM474239(2-(2,6-difluorobenzyl)-8-(2-(difluoromethoxy) pyri...)
Affinity DataIC50: 5.5nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474229BDBM474229(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50: 5.5nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474231BDBM474231(6-[[5-amino-7-(4-fluorophenyl)-8-[imidazo[1,2-a] p...)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474226BDBM474226(5-(5-amino-2-(2,6-difluorobenzyl)-7-(oxazol-2- y1)...)
Affinity DataIC50: 6.80nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474236BDBM474236(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50: 7.20nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474227BDBM474227(5-[5-amino-2-[(2,6-difluorophenyl)methyl]-7-(2 H-1...)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474240BDBM474240(8-(2-(difluoromethoxy)pyridin-4-yl)-2-((3-fluoro p...)
Affinity DataIC50: 8.30nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474224BDBM474224(5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] me...)
Affinity DataIC50: 8.70nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474226BDBM474226(5-(5-amino-2-(2,6-difluorobenzyl)-7-(oxazol-2- y1)...)
Affinity DataIC50: 12nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474225BDBM474225(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (ox...)
Affinity DataIC50: 20nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474240BDBM474240(8-(2-(difluoromethoxy)pyridin-4-yl)-2-((3-fluoro p...)
Affinity DataIC50: 21nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474225BDBM474225(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (ox...)
Affinity DataIC50: 43nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474236BDBM474236(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50: 46nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474241BDBM474241(2-[(3-fluoropyridin-2-yl)methyl]-8-[imidazo[l,2- a...)
Affinity DataIC50: 52nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474228BDBM474228(2-((3-fluoropyridin-2-yl)methyl)-8-(imidazo[l,2- a...)
Affinity DataIC50: 137nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474224BDBM474224(5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] me...)
Affinity DataIC50: 1.07E+3nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474221BDBM474221(8-(2,6-dimethylpyridin-4-yl)-7-(4-fluoropheny1)- 2...)
Affinity DataIC50: 2.87E+3nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Dizal (Jiangsu) Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 474223BDBM474223(2-(2,6-difluorobenzyl)-8-(2-(dimethylamino) pyridi...)
Affinity DataIC50: 4.77E+3nMAssay Description:Binding affinity and specificities of the compounds against different subtype of human adenosine receptors (hA1, hA2A, hA2B and hA3) were characteriz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2023
Entry Details
US Patent

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