Affinity DataKi: 500nMAssay Description:Displacement of radiolabeled PDBU from PKC in rat forebrainMore data for this Ligand-Target Pair
Affinity DataIC50: 35.2nMAssay Description:Displacement of radiolabeled PDBU from PKC in rat forebrainMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of substance P receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of substance P receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2.88E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 3.54E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >7.00E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7.32E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+4nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+5nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+5nMAssay Description:Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against recombinant human adenylate cyclase 5 expressed in HEK293 cells.More data for this Ligand-Target Pair