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Found 14 Enz. Inhib. hit(s) with all data for entry = 50044559
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020725(CHEMBL3291439)
Affinity DataIC50:  260nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020716(CHEMBL3286447)
Affinity DataIC50:  360nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020717(CHEMBL3291433)
Affinity DataIC50:  440nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020724(CHEMBL3291438)
Affinity DataIC50:  550nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020723(CHEMBL3291437)
Affinity DataIC50:  570nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020722(CHEMBL3291436)
Affinity DataIC50:  610nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020721(CHEMBL3291435)
Affinity DataIC50:  780nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020720(CHEMBL3291434)
Affinity DataIC50:  810nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020715(CHEMBL3291222)
Affinity DataIC50:  840nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020726(CHEMBL3291221)
Affinity DataIC50:  890nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020727(CHEMBL3291220)
Affinity DataIC50:  910nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020728(CHEMBL3291219)
Affinity DataIC50:  940nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020729(CHEMBL3291218)
Affinity DataIC50:  970nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50020714(CHEMBL3291217)
Affinity DataIC50:  990nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed