Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 3242
TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395229BDBM395229(US10308628, Compound 1)
Affinity DataKi:  7nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395233BDBM395233(US10308628, Compound 5)
Affinity DataKi:  9nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395230BDBM395230(US10308628, Compound 2)
Affinity DataKi:  9nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395232BDBM395232(US10308628, Compound 4)
Affinity DataKi:  15nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395231BDBM395231(US10308628, Compound 3)
Affinity DataKi:  17nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395238BDBM395238(US10308628, Compound 10)
Affinity DataKi:  21nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395237BDBM395237(US10308628, Compound 9)
Affinity DataKi:  23nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395234BDBM395234(US10308628, Compound 6)
Affinity DataKi:  26nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395236BDBM395236(US10308628, Compound 8)
Affinity DataKi:  30nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Novartis

US Patent
LigandChemical structure of BindingDB Monomer ID 395235BDBM395235(US10308628, Compound 7)
Affinity DataKi:  50nMAssay Description:15 μL of [125I]CGP 42112A, at a final concentration of 0.05 nM was added to wells of assay plate.Membranes were dispersed using a 21 gauge needl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent