Compile Data Set for Download or QSAR
Report error Found 565 Enz. Inhib. hit(s) with all data for entry = 10510
LigandChemical structure of BindingDB Monomer ID 542562BDBM542562((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0140nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542561BDBM542561((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0210nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542679BDBM542679((1 S,3′R,6′R,7′S, 8′E,15&#...)
Affinity DataKi:  0.0350nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542690BDBM542690((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0410nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542691BDBM542691((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0420nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542678BDBM542678((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0420nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542558BDBM542558((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0430nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542582BDBM542582(US11274105, Example 72)
Affinity DataKi:  0.0450nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514220BDBM50514220(CHEMBL4535151 | US11274105, Example 188)
Affinity DataKi:  0.0450nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542705BDBM542705((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0470nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542706BDBM542706((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0470nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514222BDBM50514222(CHEMBL4580244 | US11274105, Example 193)
Affinity DataKi:  0.0480nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542693BDBM542693((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0500nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542701BDBM542701((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0510nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514203BDBM50514203(CHEMBL4593361 | US11274105, Example 6)
Affinity DataKi:  0.0530nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542545BDBM542545((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0530nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542526BDBM542526((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0540nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514199BDBM50514199(CHEMBL4553660 | US11274105, Example 182)
Affinity DataKi:  0.0560nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542557BDBM542557((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0560nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542700BDBM542700((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0570nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514202BDBM50514202(CHEMBL4446369 | US11274105, Example 179)
Affinity DataKi:  0.0620nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 542525BDBM542525((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0650nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542681BDBM542681((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0660nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542579BDBM542579(US11274105, Example 70 | (3R,6R,7S,11R,17R,24S)-6&...)
Affinity DataKi:  0.0660nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542677BDBM542677((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0670nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542556BDBM542556((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0680nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542559BDBM542559((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0710nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542676BDBM542676((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0710nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542704BDBM542704((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0710nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542687BDBM542687((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0730nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542637BDBM542637((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0750nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542588BDBM542588((3R,6R,7S,11S,17R,24S)-6′-CHLORO-17-HYDROXY-...)
Affinity DataKi:  0.0810nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542527BDBM542527((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0810nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542674BDBM542674((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0860nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542538BDBM542538((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0880nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514215BDBM50514215(CHEMBL4577379 | US11274105, Example 4)
Affinity DataKi:  0.0890nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542656BDBM542656((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0900nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542547BDBM542547((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0920nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542589BDBM542589((3R,6R,7S,11S,17R,24S)-6′-CHLORO-N-(CYCLOPRO...)
Affinity DataKi:  0.0920nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542598BDBM542598((1S,3′R,6′R,7′S,8′E,16R...)
Affinity DataKi:  0.0930nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542560BDBM542560((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0930nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542528BDBM542528((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0930nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542712BDBM542712(US11274105, Example 209b | (1S,3′R,6′R...)
Affinity DataKi:  0.0960nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 542622BDBM542622(US11274105, Example 112)
Affinity DataKi:  0.0970nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514216BDBM50514216(CHEMBL4528051 | US11274105, Example 5)
Affinity DataKi:  0.0970nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 542657BDBM542657((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataKi:  0.0980nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514214BDBM50514214(CHEMBL4542646 | US11274105, Example 41)
Affinity DataKi:  0.0990nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 542562BDBM542562((1S,3′R,6′R,7′S,8′E,15R...)
Affinity DataIC50: 0.100nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514219BDBM50514219(CHEMBL4438074 | US11274105, Example 181)
Affinity DataKi:  0.103nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50514218BDBM50514218(CHEMBL4539543 | US11274105, Example 197)
Affinity DataKi:  0.104nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
US Patent

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