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Found 135 with Last Name = 'norrholm' and Initial = 'sd'
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50017701(3-Isobutyl-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)
Affinity DataKi:  41nMAssay Description:Inhibition of [3H]5HT uptake at SERT in rat brain hippocampal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM50171941((2R,6S)-1-Methyl-2,6-bis-((E)-styryl)-piperidine |...)
Affinity DataKi:  43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50192903(8R-hydroxylobel-9-ene | CHEMBL425617)
Affinity DataKi:  44nMAssay Description:Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM50080827((2R,6S)-1-Methyl-2,6-diphenethyl-piperidine | (2S,...)
Affinity DataKi:  97nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM50171941((2R,6S)-1-Methyl-2,6-bis-((E)-styryl)-piperidine |...)
Affinity DataKi:  277nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM86207(CAS_50-36-2 | COCAINE | NSC_446220)
Affinity DataKi:  469nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM50080827((2R,6S)-1-Methyl-2,6-diphenethyl-piperidine | (2S,...)
Affinity DataKi:  530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171947((2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-1-yl-ethyl)...)
Affinity DataKi:  630nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171947((2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-1-yl-ethyl)...)
Affinity DataKi:  630nMAssay Description:Binding affinity to VMAT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50192903(8R-hydroxylobel-9-ene | CHEMBL425617)
Affinity DataKi:  860nMAssay Description:Inhibition of [3H]5HT uptake at SERT in rat brain hippocampal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50080827((2R,6S)-1-Methyl-2,6-diphenethyl-piperidine | (2S,...)
Affinity DataKi:  970nMAssay Description:Binding affinity to VMAT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50080827((2R,6S)-1-Methyl-2,6-diphenethyl-piperidine | (2S,...)
Affinity DataKi:  970nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309686((2S,6S,2R)-2-[6-(2-Isobutyryloxy-2-phenylethyl)-1-...)
Affinity DataKi:  1.06E+3nMAssay Description:Inhibition of [3H]5HT uptake at SERT in rat brain hippocampal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309685((2S,6S,2R)-2-[6-(2-Toluyloxy-2-phenylethyl)-1-meth...)
Affinity DataKi:  1.51E+3nMAssay Description:Inhibition of [3H]5HT uptake at SERT in rat brain hippocampal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309687((2S,6S,2R)-2-[6-(2-Benzoyloxy-2-phenylethyl)-1-met...)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309685((2S,6S,2R)-2-[6-(2-Toluyloxy-2-phenylethyl)-1-meth...)
Affinity DataKi:  1.76E+3nMAssay Description:Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM50080827((2R,6S)-1-Methyl-2,6-diphenethyl-piperidine | (2S,...)
Affinity DataKi:  1.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM50047021(2-(6-(2-hydroxy-2-phenylethyl)-1-methylpiperidin-2...)
Affinity DataKi:  1.87E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM50171941((2R,6S)-1-Methyl-2,6-bis-((E)-styryl)-piperidine |...)
Affinity DataKi:  1.89E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309684((2S,6S,2R)-2-[6-(2-Butylsulfonyloxy-2-phenylethyl)...)
Affinity DataKi:  1.98E+3nMAssay Description:Displacement of [3HDTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171940((2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-2-yl-ethyl)...)
Affinity DataKi:  2.03E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309688((2S,6S,2R)-2-[6-(2-Anisoyloxy-2-phenylethyl)-1-met...)
Affinity DataKi:  2.04E+3nMAssay Description:Inhibition of [3H]5HT uptake at SERT in rat brain hippocampal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309685((2S,6S,2R)-2-[6-(2-Toluyloxy-2-phenylethyl)-1-meth...)
Affinity DataKi:  2.06E+3nMAssay Description:Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309687((2S,6S,2R)-2-[6-(2-Benzoyloxy-2-phenylethyl)-1-met...)
Affinity DataKi:  2.07E+3nMAssay Description:Inhibition of [3H]5HT uptake at SERT in rat brain hippocampal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171951((2R,6S)-2-((E)-Styryl)-6-styryl-piperidine | CHEMB...)
Affinity DataKi:  2.08E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309672((2S,6S,2R)-2-[6-(2-Isopropylsulfonyloxy-2-phenylet...)
Affinity DataKi:  2.09E+3nMAssay Description:Displacement of [3HDTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309687((2S,6S,2R)-2-[6-(2-Benzoyloxy-2-phenylethyl)-1-met...)
Affinity DataKi:  2.31E+3nMAssay Description:Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171953((2R,6S)-2,6-Diphenethyl-piperidine | CHEMBL192329 ...)
Affinity DataKi:  2.31E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171937(CHEMBL190725 | Methyl-bis-((E)-3-phenyl-allyl)-ami...)
Affinity DataKi:  2.37E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309686((2S,6S,2R)-2-[6-(2-Isobutyryloxy-2-phenylethyl)-1-...)
Affinity DataKi:  2.38E+3nMAssay Description:Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171952((2S,6S)-1,1-Dimethyl-2,6-diphenethyl-piperidinium;...)
Affinity DataKi:  2.39E+3nMAssay Description:Inhibition of 3 nM [3H]-MLA binding to Nicotinic acetylcholine receptor alpha7 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University of Kentucky

Curated by PDSP Ki Database
LigandPNGBDBM86207(CAS_50-36-2 | COCAINE | NSC_446220)
Affinity DataKi:  2.42E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309673((2S,6S,2R)-2-[6-(2-(2-Naphthalene)-sulfonyloxy-2-p...)
Affinity DataKi:  2.48E+3nMAssay Description:Displacement of [3HDTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171933((2S,6R)-1-Methyl-2-phenethyl-6-((E)-styryl)-piperi...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309686((2S,6S,2R)-2-[6-(2-Isobutyryloxy-2-phenylethyl)-1-...)
Affinity DataKi:  2.61E+3nMAssay Description:Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171946((2R,6S)-1-Methyl-2-phenethyl-6-((E)-styryl)-piperi...)
Affinity DataKi:  2.67E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50422013(LOBELINE | Lobeline Hydrochloride)
Affinity DataKi:  2.76E+3nMAssay Description:Binding affinity to VMAT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50080818((-)-lobeline | 2-(6-(2-Hydroxy-2-phenylethyl)-1-me...)
Affinity DataKi:  2.76E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309688((2S,6S,2R)-2-[6-(2-Anisoyloxy-2-phenylethyl)-1-met...)
Affinity DataKi:  2.98E+3nMAssay Description:Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309683((2S,6S,2R)-2-[6-(2-p-Fluoro-benzenesulfonyloxy-2-p...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3HDTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309671((2S,6S,2R)-2-[6-(2-(2-Thiophen)-carboxyl-2-phenyle...)
Affinity DataKi:  3.02E+3nMAssay Description:Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171930((2R,6S)-1-Methyl-2,6-diphenethyl-1,2,3,6-tetrahydr...)
Affinity DataKi:  3.02E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50080813(CHEMBL122636 | Methyl-bis-(3-phenyl-propyl)-amine)
Affinity DataKi:  3.07E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309670((2S,6S,2R)-2-[6-(2-p-Chloro-benzenesulfonyloxy-2-p...)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [3HDTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309682((2S,6S,2R)-2-[6-(2-Butyryloxy-2-phenylethyl)-1-met...)
Affinity DataKi:  3.38E+3nMAssay Description:Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309674((2S,6S,2R)-2-[6-(2-Benzenesulfonyloxy-2-phenylethy...)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3HDTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50309688((2S,6S,2R)-2-[6-(2-Anisoyloxy-2-phenylethyl)-1-met...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171934((2S,6S)-1-Methyl-6-phenethyl-2-((E)-styryl)-1,2,3,...)
Affinity DataKi:  3.84E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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