Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with Target = 'Bis(5'-adenosyl)-triphosphatase'
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350516BDBM50350516(CHEMBL1812066)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad protein hydrolytic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81576BDBM81576(AppppA analog, 6 (X=S))
Affinity DataKi:  35nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350512BDBM50350512(CHEMBL1812070)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad protein hydrolytic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350513BDBM50350513(CHEMBL1812069)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad protein hydrolytic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350514BDBM50350514(CHEMBL1812068)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad protein hydrolytic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350515BDBM50350515(CHEMBL1812067)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad protein hydrolytic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81584BDBM81584(AppppA analog, 12 (X=S))
Affinity DataKi:  40nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580671BDBM50580671(CHEMBL5083166)
Affinity DataIC50: 49nMAssay Description:Inhibition of human FHIT expressed in Escherichia coli BL21(DE3)-RIL cells using AP3A as substrate pretreated for 10 mins followed by substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580669BDBM50580669(CHEMBL5079345)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human FHIT assessed as reduction in AP3Aase activity measured after 45 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81586BDBM81586(AppppA analog, 13 (X=S))
Affinity DataKi:  65nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81590BDBM81590(AppppA analog, 15 (X=S))
Affinity DataKi:  78nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81593BDBM81593(AppppA analog, 17 (X=S))
Affinity DataKi:  110nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580669BDBM50580669(CHEMBL5079345)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580665BDBM50580665(CHEMBL5078809)
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human FHIT assessed as reduction in AP3Aase activity measured after 45 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81575BDBM81575(AppppA analog, 5 (X=S))
Affinity DataKi:  220nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81580BDBM81580(AppppA analog, 9 (X=S))
Affinity DataKi:  230nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81592BDBM81592(AppppA analog, 17 (X=O))
Affinity DataKi:  420nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81588BDBM81588(AppppA analog, 14 (X=S))
Affinity DataKi:  700nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580675BDBM50580675(CHEMBL5075611)
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81587BDBM81587(AppppA analog, 14 (X=O))
Affinity DataKi:  900nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580679BDBM50580679(CHEMBL5093727)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81574BDBM81574(AppppA analog, 5 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81589BDBM81589(AppppA analog, 15 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81583BDBM81583(AppppA analog, 12 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580672BDBM50580672(CHEMBL5078205)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580665BDBM50580665(CHEMBL5078809)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81570BDBM81570(AppppA analog, 1 (X=O))
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81571BDBM81571(AppppA analog, 2 (X=S))
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81591BDBM81591(AppppA analog, 16 (X=S))
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580667BDBM50580667(CHEMBL5069986)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81579BDBM81579(AppppA analog, 8 (X=S))
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81585BDBM81585(AppppA analog, 13 (X=O))
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81581BDBM81581(AppppA analog, 10 (X=S))
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580674BDBM50580674(CHEMBL5076149)
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580676BDBM50580676(CHEMBL5081769)
Affinity DataIC50: 3.73E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580677BDBM50580677(CHEMBL5075193)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580659BDBM50580659(CHEMBL5088775)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580678BDBM50580678(CHEMBL5093738)
Affinity DataIC50: 4.24E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580673BDBM50580673(CHEMBL1520857)
Affinity DataIC50: 4.66E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81577BDBM81577(AppppA analog, 6 (X=O))
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580668BDBM50580668(CHEMBL1444825)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81582BDBM81582(AppppA analog, 11 (X=S))
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580664BDBM50580664(CHEMBL5077048)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580670BDBM50580670(CHEMBL5092878)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580663BDBM50580663(CHEMBL5083554)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580671BDBM50580671(CHEMBL5083166)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580666BDBM50580666(CHEMBL5081492)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580660BDBM50580660(CHEMBL5070193)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580671BDBM50580671(CHEMBL5083166)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of recombinant human FHIT assessed as reduction in AP3Aase activity measured after 45 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBis(5'-adenosyl)-triphosphatase(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580662BDBM50580662(CHEMBL5085768)
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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