Compile Data Set for Download or QSAR
Report error Found 996 Enz. Inhib. hit(s) with Target = 'Sialidase'
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50028503BDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 0.500nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453894BDBM50453894(CHEMBL2114178)
Affinity DataIC50: 0.500nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453893BDBM50453893(CHEMBL3220445)
Affinity DataIC50: 0.500nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5000BDBM5000((3R,4R,5S)-4-Acetamido-5-amino-3-(1(S)-(2-cyclohex...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4994BDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4997BDBM4997((3R,4R,5S)-5-amino-3-[(3S)-decan-3-yloxy]-4-acetam...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4995BDBM4995((3R,4R,5S)-4-Acetamido-5-amino-3-[[(1S)-1-ethylbut...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5009BDBM5009(carbocyclic analogue 18 | (3R,4R,5S)-5-carbamimida...)
Affinity DataIC50: 2nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5015BDBM5015((3S,4R,5S)-5-amino-4-acetamido-2-fluoro-3-(pentan-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5010BDBM5010((3R,4R,5S)-4-Acetamido-5-guanidinyl-3-butoxy-1-cyc...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5227BDBM5227((3R,4R,5S)-5-amino-4-acetamido-3-[methyl(pentan-3-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4993BDBM4993((3R,4R,5S)-5-amino-3-[(2S)-butan-2-yloxy]-4-acetam...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5234BDBM5234((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-ylamino...)
Affinity DataIC50: 11nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5232BDBM5232((3R,4R,5S)-5-amino-3-(dipropylamino)-4-acetamidocy...)
Affinity DataIC50: 12nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5004BDBM5004((3R,4R,5S)-5-amino-4-acetamido-3-{[(3R)-1-phenylpe...)
Affinity DataIC50: 12nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4999BDBM4999((3R,4R,5S)-4-Acetamido-5-amino-3-(1(S)-(cyclohexyl...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5216BDBM5216((3R,4R,5S)-5-amino-3-(cyclopentyloxy)-4-acetamidoc...)
Affinity DataIC50: 22nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase-4(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50331678BDBM50331678((2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-...)
Affinity DataKi:  30nMAssay Description:Inhibition of human NEU4 using 4-MU-NANA as substrate measured every 30 seconds for 60 mins by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSialidase-1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465984BDBM50465984(CHEMBL4278858)
Affinity DataKi:  53nMAssay Description:Competitive inhibition of human His6-tagged NEU1 expressed in HEK293 cells using 4MU-NANA as substrate preincubated with substrate for 15 mins and me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278443BDBM50278443(1,3,6,7-tetrahydroxy-2-(3-methylbut-2-enyl)-8-(2-m...)
Affinity DataKi:  58nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase-4(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50331679BDBM50331679((2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-...)
Affinity DataKi:  60nMAssay Description:Inhibition of human NEU4 using 4-MU-NANA as substrate measured every 30 seconds for 60 mins by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5225BDBM5225((3R,4R,5S)-5-amino-4-acetamido-3-[methyl(propyl)am...)
Affinity DataIC50: 65nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278443BDBM50278443(1,3,6,7-tetrahydroxy-2-(3-methylbut-2-enyl)-8-(2-m...)
Affinity DataIC50: 80nMAssay Description:Inhibition of Clostridium perfringens neuraminidase by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5231BDBM5231((3R,4R,5S)-5-amino-3-[butyl(ethyl)amino]-4-acetami...)
Affinity DataIC50: 85nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5007BDBM5007((3R,4R,5S)-5-amino-4-acetamido-3-[3-(4-phenylpheny...)
Affinity DataIC50: 90nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50355214BDBM50355214(CHEMBL401566)
Affinity DataIC50: 90nMAssay Description:Inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5230BDBM5230((3R,4R,5S)-5-amino-4-acetamido-3-[ethyl(propyl)ami...)
Affinity DataIC50: 90nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175018BDBM50175018(cudraxanthone M | 4,7,8-trihydroxy-2,3,3-trimethyl...)
Affinity DataKi:  98nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5228BDBM5228((3R,4R,5S)-5-amino-4-acetamido-3-[methyl(2-phenyle...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase A(Streptococcus pneumoniae)
Korea Research Institute of Bioscience and Biotechnology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50182491BDBM50182491(CHEBI:69015 | Malabaricone C)
Affinity DataKi:  100nMAssay Description:Competitive inhibition of Streptococcus pneumoniae sialidase NanA using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5008BDBM5008((3R,4R,5S)-5-carbamimidamido-4-acetamido-3-hydroxy...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378020BDBM50378020(MACLURAXANTHONE)
Affinity DataKi:  103nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50355214BDBM50355214(CHEMBL401566)
Affinity DataKi:  110nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278443BDBM50278443(1,3,6,7-tetrahydroxy-2-(3-methylbut-2-enyl)-8-(2-m...)
Affinity DataKi:  127nMAssay Description:Apparent binding affinity at Clostridium perfringens neuraminidase by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442400BDBM50442400(AURICULASIN)
Affinity DataKi:  130nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid sodium salt hydrate as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278346BDBM50278346(Cudratricusxanthone | CHEMBL470844)
Affinity DataKi:  136nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175013BDBM50175013(cudraxanthone L | 1,3,6,7-tetrahydroxy-5-(3-methyl...)
Affinity DataKi:  138nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase-1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465993BDBM50465993(CHEMBL4290253)
Affinity DataIC50: 140nMAssay Description:Inhibition of human His6-tagged NEU1 expressed in HEK293 cells using 4MU-NANA as substrate preincubated for 15 mins followed by substrate addition an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175019BDBM50175019(cudraxanthone D | 2,3,8-trihydroxy-6-methoxy-1-(3-...)
Affinity DataKi:  143nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by Lineweaver-Burke plot and Dixon plotMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50325675BDBM50325675(smeathxanthone A | CHEMBL480158)
Affinity DataKi:  150nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50355210BDBM50355210(CHEMBL1835715)
Affinity DataKi:  160nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50355212BDBM50355212(CHEMBL1835717)
Affinity DataKi:  160nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSialidase-4(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50331678BDBM50331678((2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human NEU4 using 4-MU-NANA as substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSialidase-4(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 738185BDBM738185(US20250144172, Compound 54)
Affinity DataIC50: 160nMAssay Description:Human sialidase inhibitors may inhibit the enzymatic activity of all human sialidases, a subset of human sialidases, or one human sialidase, all in w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/9/2025
Entry Details
US Patent

TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50355212BDBM50355212(CHEMBL1835717)
Affinity DataIC50: 170nMAssay Description:Inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSialidase-1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465968BDBM50465968(CHEMBL4291908)
Affinity DataKi:  180nMAssay Description:Competitive inhibition of human His6-tagged NEU1 expressed in HEK293 cells using 4MU-NANA as substrate preincubated with substrate for 15 mins and me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5226BDBM5226((3R,4R,5S)-5-amino-3-[butyl(methyl)amino]-4-acetam...)
Affinity DataIC50: 180nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453892BDBM50453892(CHEMBL3220446)
Affinity DataIC50: 180nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175018BDBM50175018(cudraxanthone M | 4,7,8-trihydroxy-2,3,3-trimethyl...)
Affinity DataIC50: 186nMAssay Description:Inhibition of Clostridium perfringens neuraminidase by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378020BDBM50378020(MACLURAXANTHONE)
Affinity DataIC50: 186nMAssay Description:Inhibition of Clostridium perfringens neuraminidase by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
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