TargetEcdysone receptor/Protein ultraspiracle homolog(Choristoneura fumiferana)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Binding affinity to Choristoneura fumiferana EcRMore data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle(Chilo suppressalis)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to Chilo suppressalis (rice stem borer) EcRMore data for this Ligand-Target Pair
TargetEcdysone receptor/USP(Plodia interpunctella)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity to Plodia interpunctella (Indian meal moth ) EcRMore data for this Ligand-Target Pair
TargetEcdysone receptor/Gene regulation protein(Heliothis virescens)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity to Heliothis virescens (tobacco budworm) EcRMore data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle(Chironomus tentans)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to Chironomus tentans EcRMore data for this Ligand-Target Pair
TargetUltraspiracle isoform-A(Aedes aegypti)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity to Aedes aegypti EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle protein(Lucilia cuprina)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Binding affinity to Lucilia cuprina EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetProtein ultraspiracle(Drosophila melanogaster)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Binding affinity to Drosophila melanogaster EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetUltraspiracle isoform B(Leptinotarsa decemlineata)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Binding affinity to Leptinotarsa decemlineata EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 6.70E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle(Anthonomus grandis)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 1.26E+4nMAssay Description:Binding affinity to Anthonomus grandis ecdysone receptor (EcR)More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 1.68E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Binding affinity to Nezara viridula EcR10More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 2.39E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 2.51E+4nMAssay Description:Binding affinity to Nezara viridula EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 2.51E+4nMAssay Description:Binding affinity to Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 5.04E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 5.11E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetEcdysone receptor/Nuclear receptor RXR-l(Locusta migratoria)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 1.00E+5nMAssay Description:Binding affinity to Locusta migratoria ecdysone receptor (EcR)More data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle protein(Myzus persicae)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: <1.26E+5nMAssay Description:Binding affinity to Myzus persicae EcR (green peach aphid)More data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle protein(Bemisia tabaci)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: <5.01E+5nMAssay Description:Binding affinity to Bemisia tabaci (sweet potato whitefly) ecdysone receptor (EcR)More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of BCRP (unknown origin) transfected in human HEK293/R2 cells assessed as potentiation of topotecan-induced cytotoxicity measured as topot...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of BCRP (unknown origin) transfected in human HEK293/R2 cells assessed as potentiation of topotecan-induced cytotoxicity measured as topot...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of BCRP (unknown origin) transfected in human HEK293/R2 cells assessed as potentiation of topotecan-induced cytotoxicity measured as topot...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of BCRP (unknown origin) transfected in human HEK293/R2 cells assessed as potentiation of topotecan-induced cytotoxicity measured as topot...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of BCRP (unknown origin) transfected in human HEK293/R2 cells assessed as potentiation of topotecan-induced cytotoxicity measured as topot...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells assessed as reduction in cell viability after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetProtein ultraspiracle(Drosophila melanogaster)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Binding affinity to Drosophila melanogaster EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle protein(Spodoptera frugiperda)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 166nMAssay Description:Binding affinity to Spodoptera frugiperda (fall armyworm) EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle protein(Spodoptera frugiperda)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 389nMAssay Description:Binding affinity to Spodoptera frugiperda (fall armyworm) EcRMore data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle(Leptinotarsa decemlineata)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 437nMAssay Description:Binding affinity to Leptinotarsa decemlineata EcRMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 904nMAssay Description:Inhibition of BCRP in human HEK293/R2 cells assessed as reduction in cell viability after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Binding affinity to Nezara viridula EcRMore data for this Ligand-Target Pair
TargetProtein ultraspiracle(Drosophila melanogaster)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:Binding affinity to Drosophila melanogaster EcRMore data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:Binding affinity to Nezara viridula EcRMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MDR in human LCC6MDR cells assessed as reduction in cell viability after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetUltraspiracle isoform B(Leptinotarsa decemlineata)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 1.74E+3nMAssay Description:Binding affinity to Leptinotarsa decemlineata EcRMore data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
TargetUltraspiracle(Nezara viridula)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair