Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 21 hits in this display
IC50: 0.600nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: 29nMAssay Description:Inhibition of human carbonic anhydrase 2 using 4-nitrophenyl acetate as substrate after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
IC50: 52nMAssay Description:Displacement of [3H]WY 14643 from human recombinant PPARalpha receptor at 10 uM after 120 mins by scintillation counting analysis relative to controlMore data for this Ligand-Target Pair
IC50: 75nMAssay Description:Displacement of [3H]muscimol from recombinant human GABAalpha1beta2gamma2 measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
IC50: 520nMAssay Description:Inhibition of human recombinant acetylcholinesterase using acetylthiocholine as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
IC50: 8.70E+3nMAssay Description:Inhibition of human recombinant C-terminal His-tagged PHGDH (1 to 533 residues) expressed in Escherichia coli using 3-phosphoglycerate as substrateMore data for this Ligand-Target Pair
IC50: 5.77E+5nMAssay Description:Inhibition of human recombinant full-length LDHA using sodium pyruvate as substrate after 60 mins by resazurin dye-based assayMore data for this Ligand-Target Pair