Compile Data Set for Download or QSAR
Report error Found 136 of ic50 for UniProtKB: P60842
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388144BDBM50388144(CHEMBL2058177)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of eIF4A1-mediated protein synthesis in human BJAB cells assessed as inhibition of [35S]Met incorporation after 72 hr by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196926BDBM50196926(Rocaglamide | CHEMBL438139 | US10085988, Compound ...)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant full length 6xHis-tagged EIF4A1 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666748BDBM50666748(CHEMBL6177866)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant full length 6xHis-tagged EIF4A1 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540861BDBM50540861(Zotatifin | Eft226 | EFT-226)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576672BDBM50576672(CHEMBL4857096)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring highly structured 5'-UTR of c-MycMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196926BDBM50196926(Rocaglamide | CHEMBL438139 | US10085988, Compound ...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576670BDBM50576670(CHEMBL4864162)
Affinity DataIC50: 5nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring highly structured 5'-UTR of c-MycMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576669BDBM50576669(CHEMBL4855528)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring highly structured 5'-UTR of c-MycMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540861BDBM50540861(Zotatifin | Eft226 | EFT-226)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of eIF4A1 in human HAP1 cells assessed as reduction in cell proliferation incubated for 72 hrs by CellTiter-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576673BDBM50576673(CHEMBL4849769)
Affinity DataIC50: 10nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring highly structured 5'-UTR of c-MycMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576672BDBM50576672(CHEMBL4857096)
Affinity DataIC50: 11nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring short 5'-UTR of tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540861BDBM50540861(Zotatifin | Eft226 | EFT-226)
Affinity DataIC50: 14nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388144BDBM50388144(CHEMBL2058177)
Affinity DataIC50: 20nMAssay Description:Inhibition of eIF4A1-mediated protein synthesis in human BJAB cells assessed as inhibition of [35S]Met incorporation after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576670BDBM50576670(CHEMBL4864162)
Affinity DataIC50: 21nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring short 5'-UTR of tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576669BDBM50576669(CHEMBL4855528)
Affinity DataIC50: 22nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring short 5'-UTR of tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576671BDBM50576671(CHEMBL4875109)
Affinity DataIC50: 25nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring highly structured 5'-UTR of c-MycMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576673BDBM50576673(CHEMBL4849769)
Affinity DataIC50: 32nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring short 5'-UTR of tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196926BDBM50196926(Rocaglamide | CHEMBL438139 | US10085988, Compound ...)
Affinity DataIC50: 47nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50335583BDBM50335583(silvestrol | CHEMBL555196)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant full length 6xHis-tagged EIF4A1 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080528BDBM50080528(Cycloheximid | 3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2...)
Affinity DataIC50: 87nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50576671BDBM50576671(CHEMBL4875109)
Affinity DataIC50: 89nMAssay Description:Inhibition of eIF4A (unknown origin) assessed as inhibition of translation of RNA featuring short 5'-UTR of tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540861BDBM50540861(Zotatifin | Eft226 | EFT-226)
Affinity DataIC50: 92nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080528BDBM50080528(Cycloheximid | 3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2...)
Affinity DataIC50: 101nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196926BDBM50196926(Rocaglamide | CHEMBL438139 | US10085988, Compound ...)
Affinity DataIC50: 135nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080528BDBM50080528(Cycloheximid | 3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2...)
Affinity DataIC50: 142nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235738BDBM50235738(Hippuristanol)
Affinity DataIC50: 204nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235738BDBM50235738(Hippuristanol)
Affinity DataIC50: 210nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540861BDBM50540861(Zotatifin | Eft226 | EFT-226)
Affinity DataIC50: 218nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080528BDBM50080528(Cycloheximid | 3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2...)
Affinity DataIC50: 226nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196926BDBM50196926(Rocaglamide | CHEMBL438139 | US10085988, Compound ...)
Affinity DataIC50: 231nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235738BDBM50235738(Hippuristanol)
Affinity DataIC50: 369nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235738BDBM50235738(Hippuristanol)
Affinity DataIC50: 400nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235738BDBM50235738(Hippuristanol)
Affinity DataIC50: 426nMAssay Description:Inhibition of eIF4A1 in human MDA-MB-231 cells assessed as inhibition of cellular-translation incubated for 4 hrs by specific tandem sequence motif r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482563BDBM50482563(Hippurin-1 | CHEMBL449854)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482566BDBM50482566(CHEMBL1222376)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482552BDBM50482552(CHEMBL507260)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482553BDBM50482553(CHEMBL1222377)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235738BDBM50235738(Hippuristanol)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of eIF4G-induced full length recombinant human N-terminal His6/SUMO-tagged eIF4A1 RNA dependent ATPase activity expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610969BDBM50610969(CHEMBL5278302)
Affinity DataIC50: 6.58E+3nMAssay Description:Inhibition of helicase activity of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using Cy3-labele...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610969BDBM50610969(CHEMBL5278302)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610981BDBM50610981(CHEMBL5275207)
Affinity DataIC50: 8.77E+3nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482550BDBM50482550(Hippuristanol 11-One | CHEMBL1222374)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482560BDBM50482560(Hippuristanol 3-Acetate | CHEMBL1222308)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610993BDBM50610993(CHEMBL5285027)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641311BDBM50641311(CHEMBL5542372)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of EIF4A1 (unknown origin) assessed as ATP hydrolysis incubated for 1 hr in presence of ATP by malachite green assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482559BDBM50482559(CHEMBL457151)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610995BDBM50610995(CHEMBL5283331)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610950BDBM50610950(CHEMBL5277447)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610994BDBM50610994(CHEMBL5286197)
Affinity DataIC50: 2.22E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Boston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610953BDBM50610953(CHEMBL5271469)
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
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