Compile Data Set for Download or QSAR
maximum 50k data
Found 163 Enz. Inhib. hit(s) with all data for entry = 5626
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91906(Chk1_40)
Affinity DataKi:  1nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91914(Chk1_48)
Affinity DataKi:  5nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91948(Chk1_80)
Affinity DataKi:  6nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91915(Chk1_49)
Affinity DataKi:  6nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91847(Chk1_122)
Affinity DataKi:  6nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91966(Chk1_97)
Affinity DataKi:  8nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91849(Chk1_125)
Affinity DataKi:  10nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91941(Chk1_72)
Affinity DataKi:  20nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91883(Chk1_19)
Affinity DataKi:  25nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91946(Chk1_78)
Affinity DataKi:  63nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91846(Chk1_121)
Affinity DataKi:  63nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91828(Chk1_102)
Affinity DataKi:  79nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91939(Chk1_70)
Affinity DataKi:  79nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91852(Chk1_128)
Affinity DataKi:  79nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91957(Chk1_89)
Affinity DataKi:  126nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91886(Chk1_21)
Affinity DataKi:  200nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91930(Chk1_62)
Affinity DataKi:  398nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91889(Chk1_24)
Affinity DataKi:  501nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM50221567(4-(5-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazo...)
Affinity DataIC50:  0.300nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM50221567(4-(5-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazo...)
Affinity DataIC50:  0.5nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM50220753(5-(6,7-dimethoxy-1,4-dihydro-indeno[1,2-c]pyrazol-...)
Affinity DataIC50:  0.810nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91906(Chk1_40)
Affinity DataIC50:  1nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM50214577(4'-(6,7-dimethoxy-1,4-dihydro-indeno[1,2-c]pyrazol...)
Affinity DataIC50:  2nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM14826(1-[5-chloro-2-(tetrahydrofuran-3-yloxy)phenyl]-3-(...)
Affinity DataIC50:  3nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM14826(1-[5-chloro-2-(tetrahydrofuran-3-yloxy)phenyl]-3-(...)
Affinity DataIC50:  3nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91827(CHEMBL232804 | Chk1_101)
Affinity DataIC50:  4nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91830(Chk1_104)
Affinity DataIC50:  4nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM14605(1-(4-amino-5-chloro-2-methoxyphenyl)-3-(5-cyanopyr...)
Affinity DataIC50:  4nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91964(CHEMBL391449 | Chk1_95)
Affinity DataIC50:  4.40nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91827(CHEMBL232804 | Chk1_101)
Affinity DataIC50:  4.40nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91914(Chk1_48)
Affinity DataIC50:  5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91847(Chk1_122)
Affinity DataIC50:  5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM50221589(4-((6,7-dimethoxy-1,4-dihydroindeno[1,2-c]pyrazol-...)
Affinity DataIC50:  5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91866(Chk1_143)
Affinity DataIC50:  5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM14605(1-(4-amino-5-chloro-2-methoxyphenyl)-3-(5-cyanopyr...)
Affinity DataIC50:  5nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91837(Chk1_110)
Affinity DataIC50:  5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91859(Chk1_136)
Affinity DataIC50:  5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM50214559(3-(4'-hydroxy-biphenyl-4-yl)-6-methoxy-2,4-dihydro...)
Affinity DataIC50:  5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91964(CHEMBL391449 | Chk1_95)
Affinity DataIC50:  6nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91826(Chk1_100)
Affinity DataIC50:  6nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91845(Chk1_120)
Affinity DataIC50:  6nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91948(Chk1_80)
Affinity DataIC50:  6nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91838(Chk1_111)
Affinity DataIC50:  7nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91915(Chk1_49)
Affinity DataIC50:  7nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91966(Chk1_97)
Affinity DataIC50:  8nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91835(Chk1_109)
Affinity DataIC50:  9nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91851(Chk1_127)
Affinity DataIC50:  9nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91953(Chk1_85)
Affinity DataIC50:  11nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91928(Chk1_60)
Affinity DataIC50:  11nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Csar

LigandPNGBDBM91849(Chk1_125)
Affinity DataIC50:  12nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
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