Compile Data Set for Download or QSAR
Report error Found 97 Enz. Inhib. hit(s) with all data for entry = 9457
TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467268((R)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-phe...)
Affinity DataIC50: 20nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467296((S)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (2...)
Affinity DataIC50: 21nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467248(3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-phenoxy...)
Affinity DataIC50: 25nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467277((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 31nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467264((S)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-phe...)
Affinity DataIC50: 32nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467265((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2-...)
Affinity DataIC50: 33nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467138(3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-phenoxy...)
Affinity DataIC50: 36nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467138(3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-phenoxy...)
Affinity DataIC50: 36nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467292((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-phen...)
Affinity DataIC50: 37nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467272((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-phen...)
Affinity DataIC50: 40nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467288((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-phen...)
Affinity DataIC50: 40nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467315((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 42nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467311((R)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (2...)
Affinity DataIC50: 42nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467261((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (3,...)
Affinity DataIC50: 42nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467237((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-(2- ...)
Affinity DataIC50: 46nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467237((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-(2- ...)
Affinity DataIC50: 46nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467245((R)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (2...)
Affinity DataIC50: 47nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467284((S)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-phe...)
Affinity DataIC50: 50nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467253((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 58nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467293((R)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (3...)
Affinity DataIC50: 59nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467297((S)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (2...)
Affinity DataIC50: 60nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467276((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-phen...)
Affinity DataIC50: 74nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467140((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 76nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467140((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 76nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467299(3-(1-acryloylpiperidin-4-yl)-7-amino-1-(4- phenoxy...)
Affinity DataIC50: 78nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467308((S)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (3...)
Affinity DataIC50: 86nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467279((S,E)-7-amino-3-(1-(4-(dimethylamino)but-2- enoyl)...)
Affinity DataIC50: 97nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467304((S)-1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (2,6-...)
Affinity DataIC50: 100nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467280((R)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-phe...)
Affinity DataIC50: 107nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467289((R)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (2...)
Affinity DataIC50: 113nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467291(7-amino-3-((S)-1-((E)-3-((R)-1-ethylazetidin-2- yl...)
Affinity DataIC50: 123nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467294((R)-7-amino-3-(1-(but-2-ynoyl)pyrrolidin-3-yl)-1- ...)
Affinity DataIC50: 124nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467241((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-(3- ...)
Affinity DataIC50: 129nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467241((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-(3- ...)
Affinity DataIC50: 129nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467285((R)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (2...)
Affinity DataIC50: 146nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467266((R)-7-amino-3-(1-(but-2-ynoyl)pyrrolidin-3-yl)- 1-...)
Affinity DataIC50: 146nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467240(3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-(2,6-di...)
Affinity DataIC50: 147nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467246((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 147nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467240(3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-(2,6-di...)
Affinity DataIC50: 147nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467283((S,E)-7-amino-3-(1-(4-(dimethylamino)but-2- enoyl)...)
Affinity DataIC50: 151nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467303(3-(1-acryloylpiperidin-4-yl)-7-amino-1-(4-(2- fluo...)
Affinity DataIC50: 161nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467302((S)-7-amino-3-(1-(but-2-ynoyl)piperidin-3-yl)-1- (...)
Affinity DataIC50: 164nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467249((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-(4- ...)
Affinity DataIC50: 167nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467273((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 175nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467252(7-amino-3-(1-(but-2-ynoyl)pyrrolidin-3-yl)-1-(4-ph...)
Affinity DataIC50: 179nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467300((S)-3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4- (3...)
Affinity DataIC50: 181nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467256(3-(1-acryloylpyrrolidin-3-yl)-7-amino-1-(4-(2,6-di...)
Affinity DataIC50: 182nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467250((S)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4- (2,...)
Affinity DataIC50: 189nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467312((R)-3-(1-acryloylpiperidin-3-yl)-7-amino-1-(4-(2- ...)
Affinity DataIC50: 196nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM467262((S)-7-amino-3-(1-(but-2-ynoyl)pyrrolidin-3-yl)- 1-...)
Affinity DataIC50: 205nMAssay Description:MTS testing kit was purchased from Promega. The DMEM, Fetal bovine serum and Penicillin-Streptomycin were purchased from Gibco. Dimethyl sulfoxide (D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

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