Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 7203
TargetAdenosine receptor A2a(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM50011300(CHEMBL2398482 | US9133197, 2)
Affinity DataKi:  8nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181012(US9133197, 4)
Affinity DataKi:  8nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM50011301(CHEMBL2398486 | US9133197, 7)
Affinity DataKi:  12nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181014(US9133197, 6)
Affinity DataKi:  19nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181011(US9133197, 3)
Affinity DataKi:  19nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181013(US9133197, 5)
Affinity DataKi:  22nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM50011300(CHEMBL2398482 | US9133197, 2)
Affinity DataKi:  27nM ΔG°:  -43.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181010(US9133197, 1)
Affinity DataKi:  51nM ΔG°:  -41.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181010(US9133197, 1)
Affinity DataKi:  53nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181013(US9133197, 5)
Affinity DataKi:  120nM ΔG°:  -39.5kJ/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM50011301(CHEMBL2398486 | US9133197, 7)
Affinity DataKi:  197nM ΔG°:  -38.3kJ/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181014(US9133197, 6)
Affinity DataKi:  216nM ΔG°:  -38.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2016
Entry Details
US Patent