Compile Data Set for Download or QSAR
maximum 50k data
Found 62 with Last Name = 'lee' and Initial = 'yz'
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238197(CHEMBL4082885)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238209(CHEMBL4072390)
Affinity DataIC50:  39nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238195(CHEMBL4090687)
Affinity DataIC50:  45nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238198(CHEMBL4061000)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238194(CHEMBL4080388)
Affinity DataIC50:  49nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238194(CHEMBL4080388)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238197(CHEMBL4082885)
Affinity DataIC50:  53nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238199(CHEMBL4099331)
Affinity DataIC50:  54nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238200(CHEMBL4087349)
Affinity DataIC50:  56nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238203(CHEMBL4074218)
Affinity DataIC50:  57nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238210(CHEMBL4065595)
Affinity DataIC50:  59nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238201(CHEMBL4065936)
Affinity DataIC50:  66nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50400050(CHEMBL2177757 | US10793535, Cmpd ID 1 | US11191732...)
Affinity DataIC50:  81nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238209(CHEMBL4072390)
Affinity DataIC50:  87nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238210(CHEMBL4065595)
Affinity DataIC50:  92nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238194(CHEMBL4080388)
Affinity DataIC50:  102nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238205(CHEMBL4098413)
Affinity DataIC50:  102nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238198(CHEMBL4061000)
Affinity DataIC50:  148nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238195(CHEMBL4090687)
Affinity DataIC50:  151nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238201(CHEMBL4065936)
Affinity DataIC50:  177nMAssay Description:Inhibition of [3H][D-Ala2,D-Leu5]enkephalin binding to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238200(CHEMBL4087349)
Affinity DataIC50:  217nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238196(CHEMBL4069677)
Affinity DataIC50:  243nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238202(CHEMBL4087025)
Affinity DataIC50:  247nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238203(CHEMBL4074218)
Affinity DataIC50:  255nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238195(CHEMBL4090687)
Affinity DataIC50:  261nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238197(CHEMBL4082885)
Affinity DataIC50:  269nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275991(4-chlorophenyl 2-phenylethenesulfonate | CHEMBL469...)
Affinity DataIC50:  302nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238196(CHEMBL4069677)
Affinity DataIC50:  355nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238205(CHEMBL4098413)
Affinity DataIC50:  381nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276033(3-phenoxyphenyl 2-phenylethenesulfonate | CHEMBL51...)
Affinity DataIC50:  382nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238199(CHEMBL4099331)
Affinity DataIC50:  391nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275989(CHEMBL469939 | p-tolyl 2-phenylethenesulfonate)
Affinity DataIC50:  407nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276029(4-(benzyloxy)phenyl 2-phenylethenesulfonate | CHEM...)
Affinity DataIC50:  703nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276030(CHEMBL471829 | ethyl 4-(styrylsulfonyloxy)benzoate)
Affinity DataIC50:  747nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238207(CHEMBL4100814)
Affinity DataIC50:  754nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238202(CHEMBL4087025)
Affinity DataIC50:  760nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238198(CHEMBL4061000)
Affinity DataIC50:  787nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238209(CHEMBL4072390)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275988(CHEMBL469938 | naphthalen-2-yl 2-phenylethenesulfo...)
Affinity DataIC50:  1.09E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238210(CHEMBL4065595)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275990(CHEMBL467711 | m-tolyl 2-phenylethenesulfonate)
Affinity DataIC50:  1.19E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238205(CHEMBL4098413)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238201(CHEMBL4065936)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238200(CHEMBL4087349)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238207(CHEMBL4100814)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of recombinant human MCF7 cells derived His-tagged GAC (L123 to S598 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275993(4-methoxyphenyl 2-phenylethenesulfonate | CHEMBL46...)
Affinity DataIC50:  1.29E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275950(CHEMBL443343 | phenyl 2-phenylethenesulfonate)
Affinity DataIC50:  1.33E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275992(2,4,6-trichlorophenyl 2-phenylethenesulfonate | CH...)
Affinity DataIC50:  1.44E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50238199(CHEMBL4099331)
Affinity DataIC50:  1.72E+3nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276031(4-formylphenyl 2-phenylethenesulfonate | CHEMBL471...)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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