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Found 56 with Last Name = 'konkel' and Initial = 'a'
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  210nMAssay Description:Inhibition of human CYP2C19 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  210nMAssay Description:Inhibition of human CYP2C19 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50090677(4-Amino-N-(2-phenyl-2H-pyrazol-3-yl)-benzenesulfon...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human CYP2C9 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50090677(4-Amino-N-(2-phenyl-2H-pyrazol-3-yl)-benzenesulfon...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human CYP2C9 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human CYP2C19 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human CYP2C19 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human CYP2C9 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human CYP2C9 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50236897(3-(furan-2-ylmethyl)-1,8-dimethyl-1H-purine-2,6(3H...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human CYP1A2 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50236897(3-(furan-2-ylmethyl)-1,8-dimethyl-1H-purine-2,6(3H...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human CYP1A2 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of human CYP2B6 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of human CYP2B6 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human CYP2C8 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human CYP2C8 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  4.32E+4nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50:  4.32E+4nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50:  4.62E+4nMAssay Description:Inhibition of human CYP2C19 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50:  4.62E+4nMAssay Description:Inhibition of human CYP2C19 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C8 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2B6 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C9 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP1A2 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2B6 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP1A2 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C8 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2B6 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP1A2 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in supersomes using 7-benzyloxyquinoline as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C9 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C8 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C8 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2B6 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2B6 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP1A2 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2D6 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531004(CHEMBL1802692)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C19 by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531005(CHEMBL4473988)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C9 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Texas Southwestern

Curated by ChEMBL
LigandPNGBDBM50531003(CHEMBL4463477)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP2C8 by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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