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Compounds Sorted by Binding Targets per Compound

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304   310   315   323   339   369   370   371   372   373   374   375   376   377   378   380   381   383   384   
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429   443   447   515   
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • Acetylcholinesterase
  • Adenosine A1 receptor
  • Adenosine A2 receptor
  • Adenosine A2a receptor
  • Adenosine A2b receptor
  • Adenosine Receptors A2a (A2a)
  • Adenosine receptor
  • Adenosine receptor A1
  • Adenosine receptor A2a
  • Adenosine receptor A2a and A3
  • Adenosine receptor A2b
  • Adenosine receptor A3
  • Adenosine receptors; A2a & A2b
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Bile salt export pump
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Chitinase 1
  • Cholinesterases; ACHE & BCHE
  • DNA-dependent protein kinase
  • Endochitinase B1
  • Glycogen phosphorylase, muscle form
  • Guanine deaminase
  • Liver glycogen phosphorylase
  • Multidrug resistance-associated protein 4
  • Muscle glycogen phosphorylase
  • Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • Phosphodiesterase 1
  • Potassium voltage-gated channel subfamily H member 2
  • Serine-protein kinase ATM
  • Serine/threonine-protein kinase ATR
  • Sodium channel protein type I I alpha subunit
  • Twik-RElated Potassium (K+) channel 1 (TREK1)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4A
143 Ki 41 IC50 1 Kd 1 EC50
  • 1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
  • 1,3,7-trimethyl-3,7-dihydropurine-2,6-dione
  • CHEMBL113
  • Caffeine (1,3,7-trimethylxanthine)
  • caffeine
  • 15-Lipoxygenase (LoxA)
  • 3C-like proteinase
  • 3C-like proteinase (3CL-PRO)
  • 5-hydroxytryptamine receptor 6
  • Androgen receptor
  • Anti-estrogen binding site (AEBS)
  • Baculoviral IAP repeat-containing protein 2/Estrogen receptor
  • Bile salt export pump
  • Bile salt export pump (BSEP)
  • C-8 sterol isomerase
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • Cyclooxygenase
  • Cyclooxygenase-1 (COX-1)
  • Cytochrome P450 1A
  • Cytochrome P450 2B6
  • Cytochrome P450 2C19
  • Cytochrome P450 2C8
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6 (2D6)
  • Cytochrome P450 3A
  • Emopamil-binding protein-like
  • Estradiol receptor beta (ERβ)
  • Estrogen receptor
  • Estrogen-related receptor alpha
  • Estrogen-related receptor gamma
  • Lysosomal acid glucosylceramidase
  • Multidrug resistance protein 1/Multidrug resistance associated protein 1
  • Multidrug resistance-associated protein 4
  • P-glycoprotein 1
  • Phospholipase D (PLD)
  • Phospholipase D (PldA)
  • Potassium voltage-gated channel subfamily H member 2
  • Progesterone receptor
  • Sigma non-opioid intracellular receptor 1
  • Transcriptional activator protein luxR
  • streptokinase A precursor
  • ubiquitin-conjugating enzyme E2 N
15 Ki 80 IC50 1 Kd 11 EC50
  • (2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethyl)dimethylamine
  • 2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}-N,N-dimethylethanamine
  • CHEMBL83
  • FOSTRIECIN SODIUM
  • NCGC00024928
  • Nolvadex
  • Tamoxifen
  • Tamoxifen (8)
  • Tamoxifen, 7
  • cid_2733526
  • med.21724, Compound Tamoxifen
  • 5-HT3A Serotonin Receptor
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2C
  • Adrenergic Alpha
  • Alpha-1A adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • Bile salt export pump
  • Calcium channel
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • D(1A) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • Dopamine transporter
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • HTR1D
  • HTR2C
  • Histamine H1 receptor
  • Multidrug resistance-associated protein 4
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Norepinephrine Monoamine transporters
  • Norepinephrine transporter
  • Potassium voltage-gated channel subfamily H member 2
  • SLC6A3
  • Serotonin (5-HT) receptor
  • Serotonin 1B/1D receptor
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • Sodium-dependent dopamine transporter
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
  • Transporter
  • adrenergic Alpha2
127 Ki 21 IC50 1 EC50
  • 1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-2-benzofuran-5-carbonitrile
  • CHEMBL549
  • CITALOPRAM
  • CITALOPRAM HYDROBROMIDE
  • Escitalopram
  • [3H]Citalopram
  • [3H]Cytalopram
  • [3H]Escitalopram
  • [3H]Lexapro
  • ALK tyrosine kinase receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Axin-1/Glycogen synthase kinase-3 beta
  • CDK2/CycE
  • CDK2/Cyclin A/Cyclin A1
  • Cell division cycle 7-related protein kinase
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 4 (CDK4)
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-dependent kinase 7
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-activated protein kinase 2
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 14
  • PKC alpha and beta-2
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase 2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK2
  • Serine/threonine-protein kinase PLK3
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase Lck
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 3
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
  • cAMP-dependent protein kinase (PKA)
39 IC50
  • CHEMBL1094408
  • US8614220, A85B1C1Z
  • 1,3-beta-glucan synthase component GLS2
  • 5'-AMP-activated protein kinase catalytic subunit alpha-1
  • Aurora kinase A/B
  • Aurora kinase A/Targeting protein for Xklp2
  • BRAF/CRAF
  • CDK2/CycE
  • CDK4/Cyclin D3
  • CDK6/CycD3
  • CDK7/Cyclin H/MNAT1
  • Calmodulin/Proto-oncogene tyrosine-protein kinase Src
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 2 (CDK2)
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 4
  • Cyclin-dependent kinase 6
  • Cyclin-dependent kinase 7
  • Cyclin-dependent kinase 9
  • Cyclin-dependent-like kinase 5
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • High affinity nerve growth factor receptor
  • MAP kinase ERK1
  • MAP kinase-activated protein kinase 2
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • Platelet-derived growth factor receptor
  • Platelet-derived growth factor receptor beta
  • RAC-alpha serine/threonine-protein kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase pim-2
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Vascular endothelial growth factor receptor 2
39 IC50
  • US10662186, Compound 63
  • 5-HT5
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2B
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adrenergic Alpha
  • Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
  • Alpha-1A adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • Bile salt export pump
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • D(1A) dopamine receptor
  • D(2) dopamine receptor
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • HTR1D
  • HTR2B
  • HTR6
  • Histamine H1 receptor
  • Multidrug resistance-associated protein 4
  • Muscarinic acetylcholine receptor M2
  • Norepinephrine transporter
  • Serotonin (5-HT) receptor
  • Serotonin 1 (5-HT1) receptor
  • Serotonin 1B/1D receptor
  • Serotonin 2 (5-HT2) receptor
  • Serotonin 3a (5-HT3a)/3b (5-HT3b)/3c (5-HT3c)/3d (5-HT3d)/3e (5-HT3e) receptor
  • Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • Sigma non-opioid intracellular receptor 1
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
122 Ki 6 IC50 26 EC50
  • 1-(3-chlorophenyl)piperazine
  • CHEMBL478
  • m-Chlorophenylpiperazine
  • mCPP
  • AP2-associated protein kinase 1
  • Aurora kinase A/Targeting protein for Xklp2
  • BMP-2-inducible protein kinase
  • CaM kinase I alpha
  • CaM kinase I delta
  • CaM kinase I gamma
  • CaM-kinase kinase beta
  • Casein kinase I
  • Casein kinase I isoform epsilon
  • Cyclin-dependent kinase 2
  • Death-associated protein kinase 2
  • Death-associated protein kinase 3
  • Dual specificity protein kinase CLK2
  • Dual specificity protein kinase CLK4
  • Dual specificity protein kinase TTK
  • Ephrin type-A receptor 3 (EPHA3)
  • MAP kinase-interacting serine/threonine-protein kinase 2
  • MAP/microtubule affinity-regulating kinase 2
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • Phosphorylase kinase
  • Ribosomal protein S6 kinase alpha 2
  • Ribosomal protein S6 kinase alpha 5
  • Serine/threonine-protein kinase 17A
  • Serine/threonine-protein kinase 2
  • Serine/threonine-protein kinase 38-like
  • Serine/threonine-protein kinase 4 (STK4)
  • Serine/threonine-protein kinase Aurora-C
  • Serine/threonine-protein kinase GAK
  • Serine/threonine-protein kinase MST2
  • Serine/threonine-protein kinase PCTAIRE-1
  • Serine/threonine-protein kinase PLK4
  • Serine/threonine-protein kinase pim-2
  • TRAF2 and NCK-interacting protein kinase (TNIK)
  • Tyrosine-protein kinase STK16 (STK16)
  • ULK3 kinase
4 IC50 38 Kd
  • SP-600125
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2B
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adrenergic alpha1B
  • Alpha-1A adrenergic receptor
  • Alpha-1D adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • Beta-3 adrenergic receptor
  • D(1A) dopamine receptor
  • D(1B) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • D(4) dopamine receptor
  • Histamine H1 receptor
  • Histamine H2 Receptor
  • Histamine H3 receptor
  • Histamine H4 receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Muscarinic acetylcholine receptor M5
  • Serotonin (5-HT) receptor
  • Sigma non-opioid intracellular receptor 1
  • Sodium-dependent dopamine transporter
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
40 Ki
  • (4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-benzofuran-5-yl}-methanone
  • CHEMBL555146
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2B
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adrenergic alpha1B
  • Alpha-1A adrenergic receptor
  • Alpha-1D adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • Beta-3 adrenergic receptor
  • D(1A) dopamine receptor
  • D(1B) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • D(4) dopamine receptor
  • Delta-type opioid receptor
  • Histamine H1 receptor
  • Histamine H2 Receptor
  • Histamine H3 receptor
  • Histamine H4 receptor
  • Kappa-type opioid receptor
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Serotonin (5-HT) receptor
  • Sodium-dependent dopamine transporter
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
39 Ki
  • (S)-1,2-Dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-9,11-dioxa-6-aza-benzo[fg]cyclopenta[b]anthracene
  • CHEMBL179440
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adrenergic alpha1B
  • Alpha-1A adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • Beta-2 adrenergic receptor
  • D(1A) dopamine receptor
  • D(1B) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • Dopamine receptor
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • Gamma-aminobutyric acid type B receptor subunit 1
  • Glutamate receptor ionotropic, NMDA 1
  • Histamine H1 receptor
  • Kappa-type opioid receptor
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Muscarinic acetylcholine receptor M5
  • OPRD1
  • Oxytocin receptor
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • Sodium-dependent dopamine transporter
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
  • Vasopressin V1b receptor
  • Vasopressin V2 receptor
41 Ki
  • 2-amino-4-sulfobutanoic acid
  • CHEMBL191727
  • DL-homocysteic acid
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adrenergic alpha1B
  • Alpha-1A adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • D(1A) dopamine receptor
  • D(1B) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • Dopamine receptor
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • Glutamate receptor ionotropic, NMDA 1
  • Glutathione reductase
  • Histamine H1 receptor
  • Kappa-type opioid receptor
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Muscarinic acetylcholine receptor M5
  • OPRD1
  • SLC6A3
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
  • Thioredoxin reductase 1, cytoplasmic
  • Thioredoxin reductase 2, mitochondrial
  • Vasopressin V1b receptor
  • Vasopressin V2 receptor
78 Ki 4 IC50
  • CHEMBL1614664
  • Hypericin
  • Pseudohypericin
  • 40S ribosomal protein S27
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Axin-1/Glycogen synthase kinase-3 beta
  • CDK2/CycE
  • CDK2/Cyclin A/Cyclin A1
  • Cell division cycle 7-related protein kinase
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 4 (CDK4)
  • Cyclin-dependent kinase 5 regulatory subunit 1
  • Fibroblast growth factor receptor 1
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-activated protein kinase 2
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 14
  • PKC alpha and beta-2
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK2
  • Serine/threonine-protein kinase PLK3
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase Lck
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 3
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
  • cAMP-dependent protein kinase (PKA)
38 IC50
  • CHEMBL1933576
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2B
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adrenergic alpha1B
  • Alpha-1A adrenergic receptor
  • Alpha-1D adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • Beta-3 adrenergic receptor
  • D(1A) dopamine receptor
  • D(1B) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • D(4) dopamine receptor
  • Histamine H1 receptor
  • Histamine H2 Receptor
  • Histamine H3 receptor
  • Histamine H4 receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Muscarinic acetylcholine receptor M5
  • Serotonin (5-HT) receptor
  • Sigma non-opioid intracellular receptor 1
  • Sodium-dependent dopamine transporter
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
38 Ki
  • CHEMBL2031737
  • ALK tyrosine kinase receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Casein kinase II alpha/beta
  • Cell division cycle 7-related protein kinase
  • Dual specificity protein kinase TTK
  • Eukaryotic elongation factor 2 kinase
  • Focal adhesion kinase 1
  • Heat shock protein HSP 90-alpha
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-activated protein kinase 2
  • Maternal embryonic leucine zipper kinase (MELK)
  • Mitogen-activated protein kinase 1
  • Pancreatic endoplasmic reticulum kinase (PERK)
  • Platelet-derived growth factor receptor beta
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase haspin
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • heat shock 70kDa protein 8 isoform 1
37 IC50 1 Kd
  • CHEMBL2443026
  • ALK tyrosine kinase receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Casein kinase II alpha/beta
  • Cell division cycle 7-related protein kinase
  • Dual specificity protein kinase TTK
  • Eukaryotic elongation factor 2 kinase
  • Focal adhesion kinase 1
  • Heat shock protein HSP 90-alpha
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-activated protein kinase 2
  • Maternal embryonic leucine zipper kinase (MELK)
  • Mitogen-activated protein kinase 1
  • Pancreatic endoplasmic reticulum kinase (PERK)
  • Platelet-derived growth factor receptor beta
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase haspin
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • heat shock 70kDa protein 8 isoform 1
37 IC50 1 Kd
  • CHEMBL2443139
  • ALK tyrosine kinase receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Casein kinase II alpha/beta
  • Cell division cycle 7-related protein kinase
  • Dual specificity protein kinase TTK
  • Eukaryotic elongation factor 2 kinase
  • Focal adhesion kinase 1
  • Heat shock protein HSP 90-alpha
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-activated protein kinase 2
  • Maternal embryonic leucine zipper kinase (MELK)
  • Mitogen-activated protein kinase 1
  • Pancreatic endoplasmic reticulum kinase (PERK)
  • Platelet-derived growth factor receptor beta
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase haspin
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • heat shock 70kDa protein 8 isoform 1
37 IC50 1 Kd
  • CHEMBL2443138
  • ALK tyrosine kinase receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Casein kinase II alpha/beta
  • Cell division cycle 7-related protein kinase
  • Dual specificity protein kinase TTK
  • Eukaryotic elongation factor 2 kinase
  • Focal adhesion kinase 1
  • Heat shock protein HSP 90-alpha
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-activated protein kinase 2
  • Maternal embryonic leucine zipper kinase (MELK)
  • Mitogen-activated protein kinase 1
  • Pancreatic endoplasmic reticulum kinase (PERK)
  • Platelet-derived growth factor receptor beta
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase haspin
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • heat shock 70kDa protein 8 isoform 1
37 IC50 1 Kd
  • CHEMBL2443044