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Compounds Sorted by Binding Targets per Compound

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304   310   315   323   339   369   370   371   372   373   374   375   376   377   378   380   381   383   384   
385   386   388   389   390   391   392   393   394   395   397   398   401   403   404   406   408   418   427   
429   443   447   515   
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • 5-hydroxytryptamine receptor 2A
  • AGTR1
  • ATPase (Na+, K+)
  • AVPR1A
  • Adenosine Kinase (AK)
  • Adenosine kinase
  • Alpha-1A adrenergic receptor
  • Angiotensin II AT2
  • BDKRB2
  • Beta-1 adrenergic receptor
  • Beta-2 adrenergic receptor
  • Bombesin
  • CCKBR
  • CGRP
  • CHRM5
  • COX-1
  • COX-2
  • Calcium channel
  • Calcium channel (DHP)
  • Calcium release-activated calcium channel
  • Cannabinoid receptor 1
  • Cannabinoid receptor 2
  • Chloride channel, TBOB
  • D(1A) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • Dopamine D1B
  • Dopamine receptor
  • EDNRA
  • EDNRB
  • Ecto-5'-nucleotidase (e5'NT)
  • GALANIN
  • GRIA3
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • Gamma-aminobutyric acid type B receptor subunit 1
  • Glutamate receptor ionotropic, NMDA 1
  • Glutamate receptor ionotropic, kainate 1
  • HTR5A
  • HTR6
  • Histamine H1 receptor
  • Histamine H2 receptor
  • Interleukin 1-Alpha
  • Kappa-type opioid receptor
  • Melatonin
  • Monoamine Oxidase Type B (MAO-B)
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • NPY2R
  • Neurokinin 1 receptor
  • Neurokinin 2 receptor
  • Neurokinin 3 receptor
  • Neuronal acetylcholine receptor
  • Neuropeptide Y
  • Norepinephrine transporter
  • Opioid receptors; mu & delta
  • PDGF
  • PTGIR
  • Potassium Channel
  • Potassium Channel (Ca2+ dependent)
  • Renal Outer Medullary Potassium (ROMK)
  • SOMATOSTATIN
  • Serotonin (5-HT) receptor
  • Serotonin 1B/1D receptor
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • Sigma non-opioid intracellular receptor 1
  • Sodium (Site 1)
  • Sodium (Site 2)
  • Sodium-dependent dopamine transporter
  • TNF-alpha
  • Thromboxane A2 receptor
  • VIP
  • Vasopressin V2 Receptor
  • adrenergic Alpha2
77 Ki 11 IC50
  • 5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-yl)-pyrido[2,3-d]pyrimidin-4-ylamine
  • 5-(3-bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-ylamine
  • ABT-702
  • CHEMBL66089