Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- 5-hydroxytryptamine receptor 2A
- AGTR1
- ATPase (Na+, K+)
- AVPR1A
- Adenosine Kinase (AK)
- Adenosine kinase
- Alpha-1A adrenergic receptor
- Angiotensin II AT2
- BDKRB2
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Bombesin
- CCKBR
- CGRP
- CHRM5
- COX-1
- COX-2
- Calcium channel
- Calcium channel (DHP)
- Calcium release-activated calcium channel
- Cannabinoid receptor 1
- Cannabinoid receptor 2
- Chloride channel, TBOB
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- Dopamine D1B
- Dopamine receptor
- EDNRA
- EDNRB
- Ecto-5'-nucleotidase (e5'NT)
- GALANIN
- GRIA3
- Gamma-aminobutyric acid receptor subunit alpha-1
- Gamma-aminobutyric acid type B receptor subunit 1
- Glutamate receptor ionotropic, NMDA 1
- Glutamate receptor ionotropic, kainate 1
- HTR5A
- HTR6
- Histamine H1 receptor
- Histamine H2 receptor
- Interleukin 1-Alpha
- Kappa-type opioid receptor
- Melatonin
- Monoamine Oxidase Type B (MAO-B)
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- NPY2R
- Neurokinin 1 receptor
- Neurokinin 2 receptor
- Neurokinin 3 receptor
- Neuronal acetylcholine receptor
- Neuropeptide Y
- Norepinephrine transporter
- Opioid receptors; mu & delta
- PDGF
- PTGIR
- Potassium Channel
- Potassium Channel (Ca2+ dependent)
- Renal Outer Medullary Potassium (ROMK)
- SOMATOSTATIN
- Serotonin (5-HT) receptor
- Serotonin 1B/1D receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sigma non-opioid intracellular receptor 1
- Sodium (Site 1)
- Sodium (Site 2)
- Sodium-dependent dopamine transporter
- TNF-alpha
- Thromboxane A2 receptor
- VIP
- Vasopressin V2 Receptor
- adrenergic Alpha2
- 5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-yl)-pyrido[2,3-d]pyrimidin-4-ylamine
- 5-(3-bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-ylamine
- ABT-702
- CHEMBL66089